{"id":"W1898934895","doi":"10.1111/j.1476-5381.2012.02217.x","title":"Discovery of new antagonists aimed at discriminating <scp>UII</scp> and <scp>URP</scp>‐mediated biological activities: insight into <scp>UII</scp> and <scp>URP</scp> receptor activation","year":2012,"lang":"en","type":"article","venue":"British Journal of Pharmacology","topic":"Cardiovascular, Neuropeptides, and Oxidative Stress Research","field":"Medicine","cited_by":35,"is_retracted":false,"has_abstract":true,"ca_institutions":"Université de Montréal; Montreal Heart Institute; Institut National de la Recherche Scientifique","funders":"Canadian Institutes of Health Research; Armand-Frappier Foundation; Heart and Stroke Foundation of Canada","keywords":"Receptor; Chemistry; Antagonist; Cell biology; Ex vivo; Biology; Biochemistry; In vitro","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0001811704,0.0005831451,0.0006039186,0.0001440243,0.0001054516,0.0002652859,0.0003508672,0.0003621206,0.001585074],"category_scores_gemma":[0.0001618352,0.0001366667,0.0003172268,0.00013191,0.0002162364,0.0002354434,0.0001777346,0.0008932396,0.0005931805],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0002527377,"about_ca_system_score_gemma":0.000242346,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0001950252,"about_ca_topic_score_gemma":0.0004475012,"domain_scores_codex":[0.9999212,0.00001260128,0.000006382742,0.00001690818,0.00001533955,0.00002750043],"domain_scores_gemma":[0.9999141,0.00001715375,0.00001931877,0.000006508608,0.00001544252,0.00002742401],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0003694406,0.00008290794,0.0002687557,0.0001457745,0.00002060837,0.0001201418,0.0000169062,0.0001305528,0.9918686,0.0001040898,0.0001406061,0.006731683],"study_design_scores_gemma":[0.0005376321,0.006479007,0.006608218,0.00004327002,0.0001772554,0.002173805,0.00006333788,0.003395489,0.968852,0.0001331026,0.0115085,0.00002826034],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9691556,0.0125893,0.01283569,0.0002998785,0.0001151203,0.0003900965,0.0006537717,0.0001407505,0.003820007],"genre_scores_gemma":[0.9649411,0.009512845,0.01784258,0.0006327896,0.0001361651,0.000421127,0.002056315,0.00004459478,0.004412478],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.001585074,"threshold_uncertainty_score":0.005302548,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.03233815871103124,"score_gpt":0.311516204344318,"score_spread":0.2791780456332867,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}