{"id":"W1898934895","doi":"10.1111/j.1476-5381.2012.02217.x","title":"Discovery of new antagonists aimed at discriminating <scp>UII</scp> and <scp>URP</scp>‐mediated biological activities: insight into <scp>UII</scp> and <scp>URP</scp> receptor activation","year":2012,"lang":"en","type":"article","venue":"British Journal of Pharmacology","topic":"Cardiovascular, Neuropeptides, and Oxidative Stress Research","field":"Medicine","cited_by":35,"is_retracted":false,"has_abstract":true,"ca_institutions":"Université de Montréal; Montreal Heart Institute; Institut National de la Recherche Scientifique","funders":"Canadian Institutes of Health Research; Armand-Frappier Foundation; Heart and Stroke Foundation of Canada","keywords":"Receptor; Chemistry; Antagonist; Cell biology; Ex vivo; Biology; Biochemistry; In vitro","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"codex-gemma-dda1882f352a","candidate_categories":["metaresearch","metaepi_narrow"],"consensus_categories":[],"category_scores_codex":[0.002007605,0.0008244407,0.002195285,0.0008578715,0.0006305468,0.0002843259,0.0005501415,0.0006668612,0.00006101916],"category_scores_gemma":[0.01091573,0.0007853875,0.0006915918,0.0008444304,0.001564977,0.001990872,0.0008442948,0.002217986,0.00002264707],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0005027828,"about_ca_system_score_gemma":0.0005718925,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0003261935,"about_ca_topic_score_gemma":0.00004461519,"domain_scores_codex":[0.992445,0.001710773,0.001699257,0.00098612,0.001426477,0.001732392],"domain_scores_gemma":[0.9886935,0.007428868,0.001462835,0.0003362293,0.0007564265,0.001322104],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0001418813,0.0009379625,0.02695381,0.0006379301,0.001668618,0.0007858815,0.006076669,0.00001117602,0.8671485,0.00002184441,0.07731014,0.01830558],"study_design_scores_gemma":[0.01139029,0.002069576,0.1518213,0.0009667118,0.0009253219,0.005394576,0.007275647,0.00006777653,0.7252529,0.00008079414,0.09460522,0.0001499897],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9778302,0.01695367,0.000397454,0.0002197669,0.001381649,0.001123887,0.0001562868,0.00008014162,0.00185691],"genre_scores_gemma":[0.9607478,0.03153526,0.0007278637,0.0006459706,0.002968181,0.00005618928,0.0002041055,0.0001559302,0.002958703],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.1418957,"threshold_uncertainty_score":0.9994597,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.03233815871103124,"score_gpt":0.311516204344318,"score_spread":0.2791780456332867,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}