{"id":"W1965411329","doi":"10.3389/fphar.2014.00161","title":"Recent methods for measuring dopamine D3 receptor occupancy in vivo: importance for drug development","year":2014,"lang":"en","type":"review","venue":"Frontiers in Pharmacology","topic":"Neurotransmitter Receptor Influence on Behavior","field":"Neuroscience","cited_by":41,"is_retracted":false,"has_abstract":true,"ca_institutions":"University of Toronto; Centre for Addiction and Mental Health","funders":"National Institute on Drug Abuse; Canadian Institutes of Health Research; National Institutes of Health","keywords":"Dopamine receptor D3; Raclopride; Receptor; Dopamine receptor D2; D2-like receptor; Dopamine receptor; Neuroscience; Addiction; Pharmacology; Medicine; Psychology; Internal medicine","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.00531849,0.001906235,0.00178911,0.002547309,0.0003726768,0.001534352,0.001602603,0.002068527,0.00313662],"category_scores_gemma":[0.004458049,0.001427693,0.000940895,0.001893868,0.001375585,0.002152463,0.001311871,0.005486622,0.003125831],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.001888271,"about_ca_system_score_gemma":0.001258219,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.002361039,"about_ca_topic_score_gemma":0.003613348,"domain_scores_codex":[0.996036,0.001518868,0.0002219033,0.0007512585,0.001352111,0.0001198735],"domain_scores_gemma":[0.9961495,0.001661765,0.0005504348,0.000306121,0.001179164,0.000152975],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"design_other","study_design_gemma":"not_applicable","study_design_scores_codex":[0.0005528196,0.0002007173,0.002203486,0.00775182,0.0004230738,0.0003529359,0.0001780865,0.001648645,0.2830079,0.01469428,0.02572015,0.663266],"study_design_scores_gemma":[0.00009758808,0.00162705,0.007829389,0.001351971,0.0005090634,0.005774557,0.0001769431,0.005409805,0.1907924,0.01328223,0.7727721,0.0003767733],"study_design_candidate":"not_applicable","study_design_consensus":null,"genre_codex":"review","genre_gemma":"review","genre_scores_codex":[0.004206543,0.7590004,0.2188802,0.004709968,0.001981325,0.0002445675,0.0009790597,0.0007377627,0.009260159],"genre_scores_gemma":[0.02411463,0.7312378,0.2211641,0.005097574,0.00179802,0.001134308,0.001647992,0.0004351065,0.01337043],"genre_candidate":"review","genre_consensus":"review","teacher_disagreement_score":0.00531849,"threshold_uncertainty_score":0.02812719,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.110797019702356,"score_gpt":0.4316791321820635,"score_spread":0.3208821124797075,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}