{"id":"W1969866636","doi":"10.1111/j.1471-4159.2006.03840.x","title":"Binding characteristics and sensitivity to endogenous dopamine of [<sup>11</sup>C]‐(+)‐PHNO, a new agonist radiotracer for imaging the high‐affinity state of D<sub>2</sub> receptors <i>in vivo</i> using positron emission tomography","year":2006,"lang":"en","type":"article","venue":"Journal of Neurochemistry","topic":"Neurotransmitter Receptor Influence on Behavior","field":"Neuroscience","cited_by":146,"is_retracted":false,"has_abstract":true,"ca_institutions":"University of Toronto; Centre for Addiction and Mental Health","funders":"","keywords":"Raclopride; Radioligand; Agonist; Chemistry; Amphetamine; Dopamine; Dopamine receptor D3; Internal medicine; Dopamine receptor D2; Striatum; Endocrinology; Receptor; Pharmacology; Biology; Medicine; Biochemistry","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0002977455,0.0002420244,0.0002551579,0.000168945,0.0001896485,0.0004734369,0.0002806813,0.0004757661,0.001240938],"category_scores_gemma":[0.0009158772,0.0004097527,0.0001595925,0.000132984,0.000471136,0.0002196204,0.000188279,0.0003732638,0.0004601061],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0006917498,"about_ca_system_score_gemma":0.0003909781,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.01176742,"about_ca_topic_score_gemma":0.01301791,"domain_scores_codex":[0.9996771,0.00006718666,0.00001229159,0.0001205946,0.0000602042,0.00006273801],"domain_scores_gemma":[0.999589,0.0001248349,0.00006539672,0.00005004476,0.00009869356,0.00007203491],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0007047438,0.00002641743,0.002978901,0.00005130191,0.00005316627,0.00007922279,0.00009551263,0.0003077868,0.9929207,0.0001174876,0.00005359271,0.002611152],"study_design_scores_gemma":[0.00004877375,0.00171096,0.2449339,0.0000196835,0.0001680553,0.002926426,0.0002196114,0.01133106,0.7349582,0.0001680197,0.003452513,0.00006287167],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.992398,0.001263087,0.004284204,0.00004403856,0.000007782116,0.00002496938,0.0003668606,0.00002549179,0.001585528],"genre_scores_gemma":[0.9933732,0.0005877656,0.002947795,0.00006568656,0.000007193204,0.00004959313,0.0006308301,0.00004050562,0.002297501],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.01176742,"threshold_uncertainty_score":0.02339786,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.0187787917615407,"score_gpt":0.2447987855887556,"score_spread":0.2260199938272149,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}