{"id":"W1971679833","doi":"10.1111/j.1463-1326.2008.01022.x","title":"Prodrug delivery of novel PTP1B inhibitors to enhance insulin signalling","year":2009,"lang":"en","type":"article","venue":"Diabetes Obesity and Metabolism","topic":"Protein Tyrosine Phosphatases","field":"Biochemistry, Genetics and Molecular Biology","cited_by":19,"is_retracted":false,"has_abstract":true,"ca_institutions":"Women's Health Research Institute","funders":"National Institutes of Health","keywords":"Prodrug; Insulin; Pharmacology; Population; Chemistry; Endocrinology; Internal medicine; Medicine; Biology","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"codex-gemma-dda1882f352a","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0002057784,0.0001584123,0.0002343428,0.00005338377,0.00006114003,0.00001839784,0.0001561577,0.00009501556,0.000003265356],"category_scores_gemma":[0.0001421462,0.0001559542,0.00006151616,0.0001291466,0.0000511384,0.00001105657,0.0001039748,0.0000722677,0.000002842103],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.000003370288,"about_ca_system_score_gemma":0.00003477394,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0000193148,"about_ca_topic_score_gemma":0.000003922068,"domain_scores_codex":[0.9990608,0.000025749,0.0002132021,0.0003311748,0.0001219206,0.000247212],"domain_scores_gemma":[0.9994622,0.0000110686,0.00008475942,0.0002212472,0.0001044094,0.0001162589],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.00002676681,0.0001671178,0.0009644183,0.00002473013,0.00002157545,3.600439e-7,0.00004628747,0.00003951181,0.9832757,0.0004024583,0.0002352489,0.01479582],"study_design_scores_gemma":[0.0002715087,0.0001148219,0.02177702,0.0000391913,0.00002675025,3.720675e-7,0.000006718176,0.00001825696,0.9710341,0.0001204093,0.006409935,0.0001809028],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9668589,0.03195966,0.0005780113,0.0001359006,0.0000850755,0.0002600898,0.00007199648,0.00001282749,0.00003760153],"genre_scores_gemma":[0.9939506,0.0004680381,0.004534926,0.0007232948,0.0002022581,0.00001317251,0.00005249324,0.00001020371,0.00004500672],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.03149162,"threshold_uncertainty_score":0.635963,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.005600818302237525,"score_gpt":0.2266244282725026,"score_spread":0.2210236099702651,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}