{"id":"W1993878927","doi":"10.1177/0333102412466967","title":"NXN-188, a selective nNOS inhibitor and a 5-HT <sub>1B/1D</sub> receptor agonist, inhibits CGRP release in preclinical migraine models","year":2012,"lang":"en","type":"article","venue":"Cephalalgia","topic":"Migraine and Headache Studies","field":"Medicine","cited_by":56,"is_retracted":false,"has_abstract":true,"ca_institutions":"NeurAxon (Canada)","funders":"Fonden til Lægevidenskabens Fremme; Lundbeckfonden","keywords":"Calcitonin gene-related peptide; Agonist; Migraine; Medicine; Pharmacology; Sumatriptan; Receptor; 5-HT receptor; Neuroscience; Endocrinology; Serotonin; Internal medicine; Neuropeptide; Psychology","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"codex-gemma-dda1882f352a","candidate_categories":["metaepi_narrow"],"consensus_categories":[],"category_scores_codex":[0.0008144921,0.0004905144,0.0009534694,0.0002899645,0.0001846066,0.00002918632,0.0001054723,0.0003815145,0.00005728162],"category_scores_gemma":[0.001240408,0.0004345433,0.0002386904,0.0005933261,0.0002808993,0.0003785065,0.0002008993,0.000892742,0.0001320331],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0001977529,"about_ca_system_score_gemma":0.0002400435,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0001258498,"about_ca_topic_score_gemma":0.0001977912,"domain_scores_codex":[0.9968644,0.0001975356,0.0008275585,0.0007088204,0.0004040438,0.0009976291],"domain_scores_gemma":[0.9980201,0.0004539487,0.0001859293,0.0004323018,0.0002470457,0.000660703],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"not_applicable","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.003263412,0.004945598,0.1403001,0.001483902,0.0007373253,0.0001382365,0.03003417,0.000009143272,0.1857636,0.001594769,0.6210296,0.01070019],"study_design_scores_gemma":[0.05381716,0.007691496,0.3531705,0.005723832,0.002498551,0.001137824,0.00783938,0.004619327,0.4317285,0.00491371,0.1213237,0.005536049],"study_design_candidate":"not_applicable","study_design_consensus":null,"genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.982946,0.007554484,0.00006661085,0.002887609,0.0001537938,0.001171571,0.0000464473,0.0001530146,0.005020495],"genre_scores_gemma":[0.9923342,0.001032887,0.0006795057,0.00122448,0.001124065,0.0001971419,0.00006497081,0.00008125515,0.003261535],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.4997059,"threshold_uncertainty_score":0.9998106,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.03767570943829707,"score_gpt":0.3040683471999832,"score_spread":0.2663926377616861,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}