{"id":"W1996889416","doi":"10.1021/ml200084n","title":"Agonists for the Chemokine Receptor CXCR4","year":2011,"lang":"en","type":"article","venue":"ACS Medicinal Chemistry Letters","topic":"Chemokine receptors and signaling","field":"Medicine","cited_by":41,"is_retracted":false,"has_abstract":true,"ca_institutions":"Centre Hospitalier Universitaire Sainte-Justine; Université de Montréal; Université de Sherbrooke","funders":"Canadian Institutes of Health Research","keywords":"Agonist; Chimera (genetics); Chemokine receptor; Receptor; Chemokine; CXCR4; Chemistry; Partial agonist; Peptide; Chemotaxis; G protein-coupled receptor; Cell biology; Pharmacology; Biology; Biochemistry; Gene","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"codex-gemma-dda1882f352a","candidate_categories":["insufficient_payload"],"consensus_categories":[],"category_scores_codex":[0.0003440159,0.0002537293,0.0003544359,0.00002257042,0.0001543439,0.00001346779,0.0002536262,0.0001214765,0.001475775],"category_scores_gemma":[0.0002050805,0.0001673434,0.0002005538,0.0001559338,0.0002439052,0.00004149886,0.00004500542,0.0003580574,0.00002416466],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.00009898893,"about_ca_system_score_gemma":0.00007334779,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.00004186097,"about_ca_topic_score_gemma":5.151525e-7,"domain_scores_codex":[0.9985025,0.000008339425,0.0003331896,0.0003517983,0.0003787166,0.0004254503],"domain_scores_gemma":[0.9989192,0.0001852242,0.0001265708,0.0004503026,0.0001064265,0.000212198],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0003462985,0.00007326104,0.001280228,0.0002721486,0.0001583736,0.00002285035,0.0006122269,4.895722e-7,0.9417027,0.00001079272,0.0517943,0.003726316],"study_design_scores_gemma":[0.001807511,0.00006473238,0.0005494865,0.0001644826,0.0002918185,0.0001804518,0.0003799361,0.00004798283,0.9231874,0.00002042189,0.07309528,0.0002104832],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9708661,0.0006963878,0.001696341,0.02110011,0.0004526605,0.0005229344,0.00001291383,0.0001203026,0.004532265],"genre_scores_gemma":[0.9879943,0.0000877858,0.001605749,0.006352809,0.002453143,0.0001037481,0.00009523722,0.00005594701,0.001251334],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.02130098,"threshold_uncertainty_score":0.999437,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.03507979467089059,"score_gpt":0.2537756671876958,"score_spread":0.2186958725168052,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}