{"id":"W2013333057","doi":"10.1038/sj.npp.1300983","title":"Dissociation between In Vivo Occupancy and Functional Antagonism of Dopamine D2 Receptors: Comparing Aripiprazole to Other Antipsychotics in Animal Models","year":2005,"lang":"en","type":"article","venue":"Neuropsychopharmacology","topic":"Neurotransmitter Receptor Influence on Behavior","field":"Neuroscience","cited_by":194,"is_retracted":false,"has_abstract":false,"ca_institutions":"University of Toronto; Centre for Addiction and Mental Health","funders":"Canadian Institutes of Health Research; Eli Lilly and Company","keywords":"Aripiprazole; Pharmacology; Antagonism; Dopamine; Dopamine receptor D2; In vivo; Dopamine receptor; Receptor; Occupancy; Psychology; Neuroscience; Chemistry; Medicine; Internal medicine; Biology; Psychiatry; Schizophrenia (object-oriented programming)","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0006976859,0.000935004,0.001249743,0.000440797,0.000449598,0.001077914,0.0007451479,0.000821472,0.002394365],"category_scores_gemma":[0.0009503646,0.000911997,0.0006766849,0.0002627103,0.001403316,0.001756056,0.0002419607,0.003080948,0.0005958115],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.001030994,"about_ca_system_score_gemma":0.0009247172,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.003514112,"about_ca_topic_score_gemma":0.01013172,"domain_scores_codex":[0.9994224,0.000195862,0.00004248626,0.00008633274,0.0001041666,0.0001487546],"domain_scores_gemma":[0.9992925,0.000162433,0.0001532929,0.0001507081,0.00006024605,0.000180796],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.006961105,0.0005050544,0.0003998671,0.00009733456,0.00009579619,0.00005751316,0.00006786796,0.000209063,0.9867249,0.0006163357,0.0002470964,0.004018115],"study_design_scores_gemma":[0.00067855,0.01830238,0.009325985,0.00002414751,0.0002514338,0.0007725265,0.0002980729,0.004858671,0.9619836,0.0007694146,0.002677314,0.00005802169],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9866085,0.002015428,0.007056061,0.0007283155,0.0001700786,0.00009183738,0.0008173441,0.0001600565,0.002352535],"genre_scores_gemma":[0.9876612,0.002665308,0.00457111,0.0002196737,0.00008214606,0.0001847176,0.001056016,0.0001144848,0.003445212],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.003514112,"threshold_uncertainty_score":0.00800997,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.06062534332914986,"score_gpt":0.3361579621093991,"score_spread":0.2755326187802492,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}