{"id":"W2023243427","doi":"10.1074/jbc.m202723200","title":"Threonine 308 within a Putative Casein Kinase 2 Site of the Cytoplasmic Tail of Leukotriene B4 Receptor (BLT1) Is Crucial for Ligand-induced, G-protein-coupled Receptor-specific Kinase 6-mediated Desensitization","year":2002,"lang":"en","type":"article","venue":"Journal of Biological Chemistry","topic":"Receptor Mechanisms and Signaling","field":"Biochemistry, Genetics and Molecular Biology","cited_by":55,"is_retracted":false,"has_abstract":true,"ca_institutions":"Université de Sherbrooke","funders":"","keywords":"Desensitization (medicine); Receptor; Casein kinase 2; Homologous desensitization; Chemistry; Threonine; Ligand (biochemistry); Protein kinase A; G protein-coupled receptor kinase; Leukotriene receptor; Protein kinase C; Kinase; Biochemistry; G protein-coupled receptor; Cell biology; Biology; Mitogen-activated protein kinase kinase; Phosphorylation; Antagonist; Serine","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0001063783,0.0004850345,0.0003187687,0.0001407355,0.0002194504,0.0003050594,0.0002231203,0.0003513616,0.002454862],"category_scores_gemma":[0.0001616384,0.0001501236,0.0004710446,0.0001492173,0.0002067274,0.0002070043,0.0001941744,0.0004453645,0.001346392],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0005569715,"about_ca_system_score_gemma":0.00024576,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0005788507,"about_ca_topic_score_gemma":0.0006257655,"domain_scores_codex":[0.9998926,0.00001978999,0.00001103142,0.00002930251,0.00002076712,0.0000264471],"domain_scores_gemma":[0.9998999,0.00001145402,0.00004868681,0.000006723872,0.000008297751,0.00002502175],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.000425293,0.00001830094,0.0002902644,0.00006892195,0.000007821383,0.0002152126,0.00001036976,0.00009221931,0.9981143,0.0001074016,0.00004660113,0.0006032895],"study_design_scores_gemma":[0.0001197311,0.0003723774,0.02494597,0.00002570973,0.0000558117,0.002288402,0.00005379945,0.001528452,0.965063,0.0001349058,0.005392381,0.00001955419],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9947447,0.00198073,0.001890036,0.0001183415,0.00004398939,0.00003081986,0.0005389161,0.00005410767,0.0005983958],"genre_scores_gemma":[0.9923756,0.001341922,0.001693433,0.0000977359,0.0000209321,0.00004601464,0.002186992,0.00002490086,0.002212557],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.002454862,"threshold_uncertainty_score":0.008212268,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.02774688687374655,"score_gpt":0.2353714860456715,"score_spread":0.207624599171925,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}