{"id":"W2025378764","doi":"10.1002/ddr.10301","title":"Proteinase‐activated receptors: Tethered ligands and receptor‐activating peptides","year":2003,"lang":"en","type":"article","venue":"Drug Development Research","topic":"Blood Coagulation and Thrombosis Mechanisms","field":"Medicine","cited_by":7,"is_retracted":false,"has_abstract":true,"ca_institutions":"University of Calgary","funders":"Canadian Institutes of Health Research; Servier; Kidney Foundation of Canada","keywords":"Receptor; Proteolysis; G protein-coupled receptor; Protease-activated receptor; Biochemistry; Ligand (biochemistry); Cell biology; Chemistry; Enzyme-linked receptor; Peptide sequence; Signal transduction; 5-HT5A receptor; Extracellular; Biology; Functional selectivity; Enzyme; Immunology","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0001904825,0.0003133693,0.0002651921,0.0002455668,0.0001147965,0.0006488755,0.0002962637,0.0008581795,0.003915389],"category_scores_gemma":[0.000179084,0.0001637374,0.0001426912,0.0001731088,0.0003940511,0.0009092717,0.0003170212,0.0006018078,0.001355905],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0004523816,"about_ca_system_score_gemma":0.0001486374,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0001368654,"about_ca_topic_score_gemma":0.0001978419,"domain_scores_codex":[0.9998591,0.00003783422,0.000008644623,0.00002110733,0.00004865475,0.00002458377],"domain_scores_gemma":[0.9999155,0.00003297405,0.00001827379,0.000004688089,0.000006048173,0.00002254486],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.001028346,0.0001370211,0.0003365154,0.001191201,0.0000370842,0.002155763,0.0001649567,0.001066459,0.8639804,0.01875751,0.002758901,0.108386],"study_design_scores_gemma":[0.0007440206,0.002793694,0.004954211,0.000271938,0.0001521298,0.02116261,0.0002001301,0.004941565,0.7010038,0.01412229,0.249561,0.00009267272],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"review","genre_gemma":"empirical","genre_scores_codex":[0.3795335,0.5624678,0.02713524,0.004181001,0.0008458699,0.0001512422,0.0002900306,0.0004104133,0.02498489],"genre_scores_gemma":[0.7855805,0.1480397,0.01425871,0.001808189,0.0007271808,0.0001047475,0.0003404607,0.00003102821,0.04910965],"genre_candidate":"empirical","genre_consensus":null,"teacher_disagreement_score":0.003915389,"threshold_uncertainty_score":0.0130983,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.07557279785949038,"score_gpt":0.3492024730517636,"score_spread":0.2736296751922732,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}