{"id":"W2025383208","doi":"10.1016/j.peptides.2008.12.018","title":"Novel kinin B1 receptor agonists with improved pharmacological profiles","year":2008,"lang":"en","type":"article","venue":"Peptides","topic":"Coagulation, Bradykinin, Polyphosphates, and Angioedema","field":"Medicine","cited_by":30,"is_retracted":false,"has_abstract":false,"ca_institutions":"Université de Sherbrooke","funders":"","keywords":"Kinin; B2 receptor; Receptor; Agonist; Pharmacology; Chemistry; Internal medicine; Endocrinology; Biology; Medicine; Bradykinin","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"codex-gemma-dda1882f352a","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0001101028,0.0002294895,0.0003511227,0.00006816388,0.0002115524,0.00001992722,0.0001008169,0.00009827271,0.0006668486],"category_scores_gemma":[0.00008149348,0.0001623554,0.0001094109,0.0001988398,0.0002673094,0.0001190858,0.00003764883,0.0001707863,0.0001186075],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.00005431939,"about_ca_system_score_gemma":0.0001745117,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0001041918,"about_ca_topic_score_gemma":0.00001465507,"domain_scores_codex":[0.9987144,0.00001997305,0.0002756371,0.0003657114,0.0002595532,0.0003646764],"domain_scores_gemma":[0.9992565,0.00009064995,0.0001108447,0.0001913727,0.0001342651,0.0002163998],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"observational","study_design_scores_codex":[0.001487777,0.001114404,0.2188287,0.0001212952,0.0003353647,0.0001280645,0.001570661,0.00001710825,0.744066,0.0005236585,0.02310224,0.008704727],"study_design_scores_gemma":[0.007739821,0.001769023,0.6212639,0.0002316007,0.0002868065,0.0007392298,0.0003061946,0.001244541,0.3134068,0.0000458835,0.05222822,0.0007379687],"study_design_candidate":"bench_or_experimental","study_design_consensus":null,"genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9941968,0.000580446,0.0002886855,0.001312139,0.0002143843,0.0005253352,0.00002144551,0.0002591895,0.00260158],"genre_scores_gemma":[0.9808297,0.0001199034,0.009868857,0.0007822512,0.0006441835,0.00007550033,0.0000798119,0.00003710094,0.007562715],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.4306592,"threshold_uncertainty_score":0.7301525,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.03653884538061605,"score_gpt":0.2750774657400702,"score_spread":0.2385386203594542,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}