{"id":"W2025383208","doi":"10.1016/j.peptides.2008.12.018","title":"Novel kinin B1 receptor agonists with improved pharmacological profiles","year":2008,"lang":"en","type":"article","venue":"Peptides","topic":"Coagulation, Bradykinin, Polyphosphates, and Angioedema","field":"Medicine","cited_by":30,"is_retracted":false,"has_abstract":false,"ca_institutions":"Université de Sherbrooke","funders":"","keywords":"Kinin; B2 receptor; Receptor; Agonist; Pharmacology; Chemistry; Internal medicine; Endocrinology; Biology; Medicine; Bradykinin","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0003202454,0.000416875,0.0005906229,0.0002390455,0.0001575388,0.00038472,0.0002659578,0.0003819078,0.00242077],"category_scores_gemma":[0.0002241779,0.0001486168,0.0002023375,0.0001147921,0.000173962,0.0004078022,0.0001849931,0.0007870537,0.0005352675],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0001501544,"about_ca_system_score_gemma":0.0001247532,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0001242727,"about_ca_topic_score_gemma":0.0004122269,"domain_scores_codex":[0.9999149,0.00002389222,0.000007265718,0.0000107297,0.00001485611,0.00002828955],"domain_scores_gemma":[0.9999284,0.0000255528,0.00001156658,0.000005077845,0.000008462248,0.000021019],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.004896261,0.000974449,0.0005462354,0.0007435697,0.0001025039,0.001141593,0.0001762401,0.0008765793,0.8560563,0.002246911,0.002102926,0.1301365],"study_design_scores_gemma":[0.01152407,0.03895387,0.02658063,0.0003281947,0.0007538961,0.01954443,0.0002598611,0.007471762,0.7990143,0.002352256,0.09296492,0.0002517397],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9300419,0.0502232,0.007496976,0.0007761024,0.000289366,0.0002650734,0.0004395987,0.0002513197,0.01021645],"genre_scores_gemma":[0.9586698,0.01998677,0.01051787,0.001039107,0.000237453,0.0002443605,0.0007733272,0.00004573201,0.008485533],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.00242077,"threshold_uncertainty_score":0.008098304,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.03653884538061605,"score_gpt":0.2750774657400702,"score_spread":0.2385386203594542,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}