{"id":"W2027698033","doi":"10.1002/syn.10232","title":"Dopamine displaces [<sup>3</sup>H]domperidone from high‐affinity sites of the dopamine D2 receptor, but not [<sup>3</sup>H]raclopride or [<sup>3</sup>H]spiperone in isotonic medium: Implications for human positron emission tomography","year":2003,"lang":"en","type":"article","venue":"Synapse","topic":"Neurotransmitter Receptor Influence on Behavior","field":"Neuroscience","cited_by":128,"is_retracted":false,"has_abstract":true,"ca_institutions":"Canada Research Chairs; University of Toronto","funders":"","keywords":"Raclopride; Spiperone; Dopamine receptor D2; Dopamine; Chemistry; Dopamine receptor; Receptor; Domperidone; Dissociation constant; Internal medicine; Endocrinology; Biology; Biochemistry; Medicine","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"codex-gemma-dda1882f352a","candidate_categories":["metaepi_narrow","insufficient_payload"],"consensus_categories":["metaepi_narrow"],"category_scores_codex":[0.001073322,0.001393154,0.00160882,0.0008059101,0.001094607,0.0002602611,0.002769816,0.0006483321,0.001119189],"category_scores_gemma":[0.001975325,0.001091668,0.0007626389,0.002583166,0.001360637,0.001065864,0.0004514707,0.00146454,0.0001006024],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.000391141,"about_ca_system_score_gemma":0.0004114133,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0007971772,"about_ca_topic_score_gemma":0.000169233,"domain_scores_codex":[0.9904132,0.001323441,0.002360899,0.002633583,0.001416897,0.001851965],"domain_scores_gemma":[0.9931707,0.00205613,0.000911239,0.002846416,0.0003680666,0.0006474158],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0008372263,0.001585986,0.03694701,0.0001693007,0.00005424982,0.00002426252,0.001316007,0.001847419,0.9551843,0.0005840458,0.000680977,0.0007691667],"study_design_scores_gemma":[0.005012568,0.001000493,0.03027541,0.0003858563,0.0002793238,0.00008159577,0.0005636686,0.0007018916,0.9560908,0.0004838389,0.003723129,0.001401412],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9897077,0.0002123462,0.000123621,0.002807219,0.0002938037,0.004008004,0.002354459,0.0003493136,0.0001434969],"genre_scores_gemma":[0.9941592,0.0002920217,0.00149471,0.0009603272,0.0002406535,0.001400987,0.0002626925,0.0002377033,0.0009516882],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.006671603,"threshold_uncertainty_score":0.9998819,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.02954203767459315,"score_gpt":0.2856384487389069,"score_spread":0.2560964110643137,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}