{"id":"W2027698033","doi":"10.1002/syn.10232","title":"Dopamine displaces [<sup>3</sup>H]domperidone from high‐affinity sites of the dopamine D2 receptor, but not [<sup>3</sup>H]raclopride or [<sup>3</sup>H]spiperone in isotonic medium: Implications for human positron emission tomography","year":2003,"lang":"en","type":"article","venue":"Synapse","topic":"Neurotransmitter Receptor Influence on Behavior","field":"Neuroscience","cited_by":128,"is_retracted":false,"has_abstract":true,"ca_institutions":"Canada Research Chairs; University of Toronto","funders":"","keywords":"Raclopride; Spiperone; Dopamine receptor D2; Dopamine; Chemistry; Dopamine receptor; Receptor; Domperidone; Dissociation constant; Internal medicine; Endocrinology; Biology; Biochemistry; Medicine","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0001512809,0.0003269553,0.0002170223,0.0001014198,0.0001615036,0.0004630108,0.0003199937,0.0003060283,0.001025783],"category_scores_gemma":[0.0001472721,0.0003064478,0.0001890208,0.0001059987,0.0002539401,0.0003019129,0.0001655336,0.0004566355,0.0003102944],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0003787888,"about_ca_system_score_gemma":0.0003501405,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.002844274,"about_ca_topic_score_gemma":0.006053194,"domain_scores_codex":[0.9999268,0.00001572409,0.000004196584,0.00001478153,0.00001271612,0.0000257866],"domain_scores_gemma":[0.9999233,0.00002114254,0.00001631428,0.00001079672,0.000007991039,0.00002037443],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0002431637,0.00001394464,0.000307332,0.00001932155,0.000007847009,0.00006598044,0.00002077234,0.00005934952,0.9981828,0.0001243791,0.00003440874,0.0009206442],"study_design_scores_gemma":[0.00002433494,0.0002042066,0.004445833,0.000002811949,0.00002004006,0.0005057166,0.00004125852,0.001252159,0.9923075,0.00007541708,0.001111424,0.000009268212],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9952005,0.0009823442,0.002483489,0.00008280479,0.00001039308,0.000008392043,0.0001224733,0.00003456327,0.001074931],"genre_scores_gemma":[0.9945052,0.0005969706,0.002922839,0.00003768079,0.000005154002,0.00001072406,0.0002238285,0.0000275164,0.001670099],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.002844274,"threshold_uncertainty_score":0.005655408,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.02954203767459315,"score_gpt":0.2856384487389069,"score_spread":0.2560964110643137,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}