{"id":"W2041535798","doi":"10.1038/nature09504","title":"Selective inhibition of BET bromodomains","year":2010,"lang":"en","type":"article","venue":"Nature","topic":"Protein Degradation and Inhibitors","field":"Biochemistry, Genetics and Molecular Biology","cited_by":4296,"is_retracted":false,"has_abstract":false,"ca_institutions":"","funders":"National Cancer Institute; Canadian Institutes of Health Research; U.S. Public Health Service; Cancer Research UK; Wellcome Trust","keywords":"Bromodomain; BRD4; Epigenetics; Chromatin; BET inhibitor; Small molecule; Histone; Fusion protein; Chemistry; Binding site; Computational biology; Acetylation; Biology; Cell biology; Cancer research; Biochemistry; Gene","routes":{"ca_aff":false,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":true},"retraction":null,"screen":null}