{"id":"W2045328857","doi":"10.1111/j.1399-3011.2005.00252.x","title":"Type and location of fluorescent probes incorporated into the potent <i>μ</i>‐opioid peptide [Dmt<sup>1</sup>]DALDA affect potency, receptor selectivity and intrinsic efficacy*","year":2005,"lang":"en","type":"article","venue":"Journal of Peptide Research","topic":"Neuropeptides and Animal Physiology","field":"Neuroscience","cited_by":12,"is_retracted":false,"has_abstract":true,"ca_institutions":"Montreal Clinical Research Institute","funders":"National Institute on Drug Abuse","keywords":"Chemistry; Agonist; μ-opioid receptor; Peptide; Tetrapeptide; Dermorphin; Receptor; Oligopeptide; Partial agonist; Stereochemistry; Biodistribution; Opioid peptide; Opioid; In vitro; Biochemistry","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0002200641,0.0004553163,0.0002400596,0.0001060347,0.0001051058,0.0003265096,0.0003102036,0.0004237791,0.000893879],"category_scores_gemma":[0.0003536012,0.0002103667,0.0001978021,0.0001083814,0.0002578576,0.000289397,0.0001096156,0.0003978966,0.0002801834],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0003208462,"about_ca_system_score_gemma":0.0001301075,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0003956178,"about_ca_topic_score_gemma":0.0004128731,"domain_scores_codex":[0.9998112,0.00003434635,0.00001683571,0.0000546097,0.00002770614,0.00005533943],"domain_scores_gemma":[0.9997004,0.0001237001,0.00008283405,0.0000311506,0.00002637548,0.00003563651],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.00009348845,0.00001274906,0.00006420154,0.00001903825,0.000002502456,0.00001308002,0.000004755257,0.0000565858,0.9991966,0.00003817932,0.000006773715,0.0004919725],"study_design_scores_gemma":[0.000007302031,0.0001621636,0.0003886979,0.000001292023,0.00001051766,0.00004970152,0.000003534974,0.0001695714,0.9989023,0.000004690826,0.000298003,0.000002302365],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9947751,0.001237364,0.002490526,0.00004086845,0.00002366832,0.00003390861,0.0001154441,0.00003927571,0.001243896],"genre_scores_gemma":[0.9947689,0.000717516,0.003543941,0.00004598481,0.000009507445,0.00002503567,0.0001563908,0.00002044446,0.0007122905],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.000893879,"threshold_uncertainty_score":0.002990365,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.04773662229322174,"score_gpt":0.3254918330813443,"score_spread":0.2777552107881225,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}