{"id":"W2051296550","doi":"10.1016/s0968-0896(00)00275-3","title":"Imidazoline-modified benzylimidazolines as h5-HT1D/1B serotonergic ligands","year":2001,"lang":"en","type":"article","venue":"Bioorganic & Medicinal Chemistry","topic":"Migraine and Headache Studies","field":"Medicine","cited_by":26,"is_retracted":false,"has_abstract":false,"ca_institutions":"IDELIX Software (Canada); Amorfix (Canada)","funders":"","keywords":"Chemistry; Imidazoline receptor; Agonist; Tryptamine; Serotonergic; Receptor; 5-HT receptor; Stereochemistry; Aromatization; Serotonin; Selectivity; Pharmacology; Biochemistry","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"codex-gemma-dda1882f352a","candidate_categories":["metaepi_narrow","insufficient_payload"],"consensus_categories":[],"category_scores_codex":[0.000346714,0.0005475084,0.0009003246,0.00009419917,0.000233736,0.00002348968,0.0002960985,0.0003858788,0.002261583],"category_scores_gemma":[0.0005093169,0.0004443497,0.0002786627,0.0006074684,0.0002905822,0.00007049492,0.0001505519,0.0006593115,0.000268877],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0001465575,"about_ca_system_score_gemma":0.0004173228,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0001358157,"about_ca_topic_score_gemma":0.00001939403,"domain_scores_codex":[0.9969868,0.00001504614,0.0007151425,0.0007007765,0.000789192,0.0007930373],"domain_scores_gemma":[0.9980518,0.00009203175,0.0001914919,0.0007386278,0.0003010361,0.0006249835],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0008091822,0.0006892974,0.009378791,0.000839525,0.000427237,0.001087079,0.001046144,0.000001449344,0.9268599,0.00009265146,0.05789803,0.0008707398],"study_design_scores_gemma":[0.007763773,0.0005259541,0.006744938,0.0007787907,0.000934845,0.00475464,0.003602726,0.0002160508,0.8905536,0.0003509847,0.08283462,0.0009390719],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9441782,0.004739391,0.00003034355,0.009556584,0.00010034,0.0003604382,0.000009633848,0.0003102635,0.04071487],"genre_scores_gemma":[0.971527,0.001979931,0.00007027598,0.002244356,0.003419915,0.00004759508,0.0001198788,0.00008023595,0.02051082],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.03630627,"threshold_uncertainty_score":0.9998008,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.02217192635021855,"score_gpt":0.3000829861579942,"score_spread":0.2779110598077757,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}