{"id":"W2052593334","doi":"10.1042/bj20080074","title":"Mutation of Trp29 of human equilibrative nucleoside transporter 1 alters affinity for coronary vasodilator drugs and nucleoside selectivity","year":2008,"lang":"en","type":"article","venue":"Biochemical Journal","topic":"Adenosine and Purinergic Signaling","field":"Biochemistry, Genetics and Molecular Biology","cited_by":23,"is_retracted":false,"has_abstract":true,"ca_institutions":"University of Alberta","funders":"Wellcome Trust","keywords":"Nucleoside; Nucleoside transporter; Chemistry; Selectivity; Transporter; Nucleoside analogue; Vasodilation; Pharmacology; Biochemistry; Gene; Biology; Internal medicine; Medicine","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0001698144,0.0005235131,0.0004398622,0.0001700872,0.0001538965,0.0002893738,0.0003588271,0.000510104,0.002079085],"category_scores_gemma":[0.0003431989,0.0001850976,0.000492501,0.0002226175,0.0003052712,0.0001973071,0.0002608951,0.0004215568,0.001096625],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0003043056,"about_ca_system_score_gemma":0.000251641,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0009204535,"about_ca_topic_score_gemma":0.00065057,"domain_scores_codex":[0.9997922,0.00005973482,0.00003294786,0.00004161617,0.00004371018,0.0000298369],"domain_scores_gemma":[0.9997168,0.00007763469,0.0001024828,0.00002832384,0.0000192053,0.00005551592],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0002561023,0.00006298831,0.0003785082,0.00002690991,0.0000210303,0.0004630409,0.00001990619,0.0005163142,0.9963163,0.0002285184,0.00007263584,0.001637747],"study_design_scores_gemma":[0.00008621849,0.0005552425,0.006246409,0.00001300471,0.0000523901,0.002862002,0.00004666307,0.007707643,0.9785372,0.0001279259,0.003729489,0.00003591935],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9948086,0.0002373828,0.003287665,0.00008892029,0.00003683495,0.00004640561,0.0005065263,0.00009640615,0.0008911884],"genre_scores_gemma":[0.9954147,0.0001830802,0.002403967,0.00007055463,0.00001348371,0.00002570964,0.0006012674,0.00007012532,0.001217059],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.002079085,"threshold_uncertainty_score":0.006955266,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.01683001522099442,"score_gpt":0.2599447936081499,"score_spread":0.2431147783871555,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}