{"id":"W2061659009","doi":"10.1021/mp800050q","title":"Effects of Monoglycerides on P-Glycoprotein: Modulation of the Activity and Expression in Caco-2 Cell Monolayers","year":2008,"lang":"en","type":"article","venue":"Molecular Pharmaceutics","topic":"Drug Transport and Resistance Mechanisms","field":"Medicine","cited_by":45,"is_retracted":false,"has_abstract":true,"ca_institutions":"University of British Columbia","funders":"","keywords":"Caco-2; Chemistry; P-glycoprotein; Apical membrane; Efflux; Biochemistry; Cell culture; Membrane; Cell; Biology; Multiple drug resistance","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0001176264,0.000264853,0.0002591012,0.00008978784,0.00011132,0.0002290601,0.0001398258,0.0002892143,0.0006258523],"category_scores_gemma":[0.0001560072,0.00009561374,0.0001637318,0.0001840006,0.0001508768,0.0002707346,0.0001772651,0.0003063345,0.000187031],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0001923294,"about_ca_system_score_gemma":0.0001389595,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0006611957,"about_ca_topic_score_gemma":0.001554152,"domain_scores_codex":[0.9998364,0.00005270998,0.0000131965,0.00002701187,0.00004684887,0.0000236915],"domain_scores_gemma":[0.9999325,0.00002165271,0.00001651161,0.000007580509,0.00001451948,0.000007097994],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0001890751,0.00001910291,0.0001025063,0.00005096273,0.000004171304,0.00004276821,0.00001864538,0.00002870431,0.998456,0.0000240618,0.00001425065,0.001049642],"study_design_scores_gemma":[0.000008010977,0.0003384078,0.002416166,0.000004439745,0.00001437276,0.0001176706,0.00002815001,0.0002486044,0.9955786,0.00001249942,0.001230404,0.000002653939],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9943491,0.003501724,0.0009627633,0.0001189107,0.00001977915,0.00002247935,0.0001575643,0.00002245059,0.0008453045],"genre_scores_gemma":[0.990303,0.004158734,0.00294286,0.0001060711,0.00001521035,0.00005256761,0.0003489212,0.00001521836,0.002057464],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.0006611957,"threshold_uncertainty_score":0.002093673,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.01289102013280416,"score_gpt":0.2584809436140839,"score_spread":0.2455899234812798,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}