{"id":"W2074117907","doi":"10.1016/j.nucmedbio.2007.08.005","title":"Dopamine D2 receptor radiotracers [11C](+)-PHNO and [3H]raclopride are indistinguishably inhibited by D2 agonists and antagonists ex vivo","year":2007,"lang":"en","type":"article","venue":"Nuclear Medicine and Biology","topic":"Neurotransmitter Receptor Influence on Behavior","field":"Neuroscience","cited_by":45,"is_retracted":false,"has_abstract":false,"ca_institutions":"Centre for Addiction and Mental Health; University of Toronto","funders":"Canadian Institutes of Health Research","keywords":"Raclopride; Dopamine receptor D2; Chemistry; Ex vivo; Dopamine; Pharmacology; Receptor; Internal medicine; Biology; Medicine; In vitro; Biochemistry","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"codex-gemma-dda1882f352a","candidate_categories":["metaepi_narrow"],"consensus_categories":[],"category_scores_codex":[0.0004854057,0.000390211,0.0005578135,0.0002369116,0.0003033947,0.00005533447,0.000225138,0.0002824893,0.0003147424],"category_scores_gemma":[0.0006582981,0.0003141086,0.00003556974,0.0003377125,0.001930296,0.0001418535,0.0001223056,0.0005108186,0.00002442081],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.00003974935,"about_ca_system_score_gemma":0.00001771746,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0001472837,"about_ca_topic_score_gemma":0.0000217176,"domain_scores_codex":[0.9974825,0.0001563309,0.0005272602,0.0009709915,0.0002097751,0.0006531673],"domain_scores_gemma":[0.9986463,0.0003538382,0.0002614212,0.0002681085,0.00005414556,0.0004161748],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"not_applicable","study_design_scores_codex":[0.0001690614,0.00005526093,0.0249694,0.00005103216,0.000006047416,0.0001013998,0.0007001443,1.653443e-8,0.9532474,0.0001063864,0.005813681,0.01478019],"study_design_scores_gemma":[0.005547362,0.002685563,0.04603827,0.0003408151,0.0001155371,0.001647741,0.001267202,0.00002769001,0.306772,0.0001303917,0.6342762,0.001151165],"study_design_candidate":"bench_or_experimental","study_design_consensus":null,"genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9933228,0.0006447297,0.000009920264,0.004274571,0.0004379289,0.0003933435,0.0000842431,0.0001469977,0.0006854761],"genre_scores_gemma":[0.9911254,0.001141503,0.0002079171,0.006919762,0.0002912751,0.000005246865,0.00001728541,0.00005722456,0.0002343582],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.6464754,"threshold_uncertainty_score":0.9999311,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.03605751440136093,"score_gpt":0.3064204526528453,"score_spread":0.2703629382514844,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}