{"id":"W2081337972","doi":"10.1152/ajpregu.90766.2008","title":"VRQ397 (CRAVKY): a novel noncompetitive V2 receptor antagonist","year":2009,"lang":"en","type":"article","venue":"American Journal of Physiology-Regulatory, Integrative and Comparative Physiology","topic":"Neuroendocrine regulation and behavior","field":"Psychology","cited_by":18,"is_retracted":false,"has_abstract":true,"ca_institutions":"McGill University; Université de Sherbrooke; Université de Montréal","funders":"Canadian Institutes of Health Research; Canada Research Chairs; Heart and Stroke Foundation of Canada","keywords":"Receptor; Vasopressin; Vasopressin receptor; Chemistry; Desmopressin; Competitive antagonist; In vivo; Arginine; Non-competitive inhibition; Antagonist; Biophysics; Biochemistry; Biology; Endocrinology; Amino acid","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0001600575,0.0006675285,0.0005857504,0.0002831047,0.0001702684,0.0003397289,0.0007238862,0.0006419941,0.001897092],"category_scores_gemma":[0.0001762601,0.0001650297,0.0003074718,0.0002848461,0.0002700991,0.0002266177,0.0002701416,0.0007435923,0.001239523],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0003709665,"about_ca_system_score_gemma":0.0003361271,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0006759595,"about_ca_topic_score_gemma":0.001122704,"domain_scores_codex":[0.9997984,0.00003267508,0.0000122551,0.00005463738,0.00004937526,0.00005273512],"domain_scores_gemma":[0.9999278,0.00001223147,0.00001824339,0.00000546363,0.00001071018,0.00002553376],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0005553706,0.0001494493,0.000222097,0.0001484339,0.00002550235,0.0002789285,0.00002278998,0.0003956768,0.9850263,0.0001934866,0.0002882675,0.01269378],"study_design_scores_gemma":[0.001944722,0.01370426,0.008308525,0.00004625733,0.000150542,0.007944803,0.00006171648,0.003780015,0.9329147,0.0001862351,0.03087868,0.00007943908],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9761722,0.01118988,0.005798296,0.0001963397,0.00009227027,0.0003194003,0.0008408182,0.0002465139,0.00514436],"genre_scores_gemma":[0.979708,0.004522494,0.007913054,0.0003241311,0.00006686343,0.0002217971,0.002346118,0.00004776154,0.004849589],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.001897092,"threshold_uncertainty_score":0.006346405,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.03294906430833582,"score_gpt":0.3412552893176512,"score_spread":0.3083062250093154,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}