{"id":"W2085971293","doi":"10.1002/cbic.201402512","title":"Identification and Characterization of a Small‐Molecule Inhibitor of Death‐Associated Protein Kinase 1","year":2014,"lang":"en","type":"article","venue":"ChemBioChem","topic":"Melanoma and MAPK Pathways","field":"Biochemistry, Genetics and Molecular Biology","cited_by":25,"is_retracted":false,"has_abstract":true,"ca_institutions":"","funders":"Ministero dello Sviluppo Economico; Strategic Research Council; Novo Nordisk; Ontario Ministry of Economic Development and Innovation; Genome Canada; Wellcome Trust; GlaxoSmithKline; Pfizer; Eli Lilly and Company","keywords":"Identification (biology); Small molecule; Chemistry; Kinase; Protein kinase A; Computational biology; Molecule; Biochemistry; Cell biology; Biology","routes":{"ca_aff":false,"ca_fund":true,"ca_venue":false,"about_ca":true,"invisible_to_affiliation_only":true},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0001240828,0.0003488619,0.0003556883,0.0001648644,0.0000963171,0.0002670685,0.0003354576,0.0002373434,0.0005895779],"category_scores_gemma":[0.0001533096,0.00009807882,0.0001938012,0.0001465159,0.0001129124,0.000194145,0.000136146,0.0003584978,0.0003396421],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.00035401,"about_ca_system_score_gemma":0.0002793031,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0004069421,"about_ca_topic_score_gemma":0.0004705072,"domain_scores_codex":[0.9999079,0.000006434901,0.000006634748,0.00001934022,0.00004178145,0.00001789811],"domain_scores_gemma":[0.9999526,0.000006341972,0.00001083655,0.000003526932,0.00001159942,0.0000151587],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.00006744308,0.00006137981,0.0001961587,0.00005166678,0.000007293827,0.00007459866,0.00000741249,0.0004936858,0.9946808,0.00006835681,0.00007877101,0.004212317],"study_design_scores_gemma":[0.00006354744,0.001165419,0.002968202,0.00000558901,0.00002891752,0.0005055789,0.000006595117,0.004292379,0.9850047,0.00004137091,0.005907877,0.000009854944],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9673459,0.008587926,0.0186761,0.0002726052,0.00004997614,0.0003239221,0.001271571,0.0001541354,0.003317945],"genre_scores_gemma":[0.9744062,0.00371687,0.01277312,0.0001428692,0.00002783978,0.0001264716,0.004169568,0.00002056598,0.004616363],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.0005895779,"threshold_uncertainty_score":0.002568483,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.00832888224529081,"score_gpt":0.2011807604510626,"score_spread":0.1928518782057718,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}