{"id":"W2086860055","doi":"10.1039/c3dt51152a","title":"A model radiopharmaceutical agent targeted to translocator protein 18 kDa (TSPO)","year":2013,"lang":"en","type":"article","venue":"Dalton Transactions","topic":"Radiopharmaceutical Chemistry and Applications","field":"Medicine","cited_by":15,"is_retracted":false,"has_abstract":true,"ca_institutions":"","funders":"Ministero dell'Università e della Ricerca; Ryerson University","keywords":"Translocator protein; Imidazopyridine; Chemistry; Ligand (biochemistry); Combinatorial chemistry; Biophysics; Biochemistry; Medicine; Biology; Receptor; Internal medicine; Inflammation","routes":{"ca_aff":false,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":true},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0001647602,0.0003728053,0.0003055006,0.0002172356,0.0001717234,0.0002300112,0.0003548933,0.0004046772,0.001178927],"category_scores_gemma":[0.0001555042,0.0001535008,0.000167488,0.0001632927,0.0003234945,0.0002068891,0.0001739243,0.0004819581,0.0005486133],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0005483543,"about_ca_system_score_gemma":0.0002507441,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.001311229,"about_ca_topic_score_gemma":0.001493654,"domain_scores_codex":[0.9998956,0.00001758133,0.000004618154,0.00003367235,0.00002633734,0.00002222001],"domain_scores_gemma":[0.9999238,0.00001426054,0.00002052366,0.000007631284,0.00001053187,0.00002332713],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.00007757456,0.00001155591,0.00003917175,0.00005780206,0.000003846628,0.00006698394,0.00001721042,0.0001482233,0.9977744,0.0002135298,0.00006394823,0.001525705],"study_design_scores_gemma":[0.00002711734,0.0003552524,0.0003907861,0.000003715875,0.00001856772,0.0004649932,0.000007437971,0.0003818761,0.9896842,0.00002326352,0.008637181,0.000005651316],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9557498,0.0072055,0.03046799,0.0004015891,0.00009980117,0.0001990274,0.0006420143,0.0003611023,0.004873211],"genre_scores_gemma":[0.9677081,0.002005312,0.0230754,0.00008945329,0.00003429561,0.00008608006,0.0006342762,0.00008317093,0.006283971],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.001311229,"threshold_uncertainty_score":0.00397855,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.05701071075540631,"score_gpt":0.3374166845065024,"score_spread":0.280405973751096,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}