{"id":"W2105607249","doi":"10.1128/aac.49.8.3483-3485.2005","title":"TAK-220, a Novel Small-Molecule CCR5 Antagonist, Has Favorable Anti-Human Immunodeficiency Virus Interactions with Other Antiretrovirals In Vitro","year":2005,"lang":"en","type":"article","venue":"Antimicrobial Agents and Chemotherapy","topic":"HIV Research and Treatment","field":"Immunology and Microbiology","cited_by":31,"is_retracted":false,"has_abstract":true,"ca_institutions":"Centre Hospitalier de l’Université de Montréal","funders":"","keywords":"CCR5 receptor antagonist; In vitro; Human immunodeficiency virus (HIV); Antagonist; Virology; Drug; Pharmacology; Virus; Medicine; Immunology; Biology; Receptor; Internal medicine; Chemokine receptor; Genetics; Inflammation","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0003141075,0.0006110318,0.0008374634,0.0002194324,0.0002375716,0.0004318377,0.0002668913,0.0002966433,0.001889371],"category_scores_gemma":[0.0003082895,0.0001948362,0.0005148005,0.0001678633,0.0002274481,0.0003523682,0.00016967,0.0008067891,0.000605554],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0001847974,"about_ca_system_score_gemma":0.0002755535,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0003800725,"about_ca_topic_score_gemma":0.0009862088,"domain_scores_codex":[0.9997358,0.00007714815,0.00002503127,0.00002570753,0.0000792982,0.00005711585],"domain_scores_gemma":[0.9998257,0.00005881792,0.00003091442,0.00001041799,0.00002307531,0.00005113592],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.002109909,0.0006888894,0.0006792847,0.0005892527,0.0001018712,0.0002330183,0.00004850114,0.0005802799,0.9666104,0.0002203452,0.0005058719,0.02763229],"study_design_scores_gemma":[0.0003959115,0.01712298,0.005992483,0.00002653727,0.0002249033,0.00238922,0.00005990237,0.001836661,0.9633321,0.00008332125,0.008494405,0.00004165377],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.969533,0.02124831,0.002500384,0.0002605713,0.0001629131,0.000103379,0.0004203811,0.000103381,0.005667648],"genre_scores_gemma":[0.9890688,0.005021404,0.002753231,0.000137537,0.00007574633,0.00005794252,0.001007162,0.00001071974,0.00186746],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.001889371,"threshold_uncertainty_score":0.006320596,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.02642900245337289,"score_gpt":0.2739155901048932,"score_spread":0.2474865876515203,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}