{"id":"W2107430154","doi":"10.1124/dmd.31.4.373","title":"Segmental Intestinal Transporters and Metabolic Enzymes on Intestinal Drug Absorption","year":2003,"lang":"en","type":"article","venue":"Drug Metabolism and Disposition","topic":"Drug Transport and Resistance Mechanisms","field":"Medicine","cited_by":70,"is_retracted":false,"has_abstract":false,"ca_institutions":"University of Toronto","funders":"","keywords":"Metabolite; Bioavailability; Glucuronidation; Small intestine; Pharmacokinetics; Transporter; Absorption (acoustics); Chemistry; Metabolism; Distribution (mathematics); Biology; Pharmacology; Biochemistry; Enzyme","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0005031452,0.0005220606,0.001122506,0.0004068009,0.0002132524,0.001136299,0.0003740086,0.0008204921,0.004891452],"category_scores_gemma":[0.0005920446,0.0002553051,0.0005159009,0.0004943994,0.0006746369,0.00190825,0.0005054194,0.0008661807,0.0007823004],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0005837968,"about_ca_system_score_gemma":0.0003097872,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0009637911,"about_ca_topic_score_gemma":0.0009575229,"domain_scores_codex":[0.9997987,0.00009901333,0.00001378992,0.00002391894,0.00003002532,0.00003447397],"domain_scores_gemma":[0.9996996,0.0001363385,0.00004740397,0.0000245626,0.0000546643,0.00003741672],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.01357618,0.0005063706,0.01838188,0.003263292,0.0005698302,0.005882287,0.0006708436,0.01185743,0.4662719,0.1168875,0.004722939,0.3574096],"study_design_scores_gemma":[0.0005807262,0.009644376,0.2277634,0.0007537754,0.001468503,0.01494199,0.0015779,0.04108295,0.4856751,0.0910656,0.1251103,0.000335312],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.62839,0.2851882,0.03478068,0.005693056,0.0002972846,0.00007517436,0.0003571446,0.000322032,0.04489642],"genre_scores_gemma":[0.9323948,0.05323016,0.002329533,0.0004066604,0.000392225,0.00002564665,0.0001589585,0.00005033011,0.01101154],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.004891452,"threshold_uncertainty_score":0.01636356,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.007315072335970585,"score_gpt":0.2238134900455058,"score_spread":0.2164984177095352,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}