{"id":"W2108223516","doi":"10.1124/jpet.110.169946","title":"Naphthalen-1-yl-(4-pentyloxynaphthalen-1-yl)methanone (SAB378), a Peripherally Restricted Cannabinoid CB1/CB2 Receptor Agonist, Inhibits Gastrointestinal Motility but Has No Effect on Experimental Colitis in Mice","year":2010,"lang":"en","type":"article","venue":"Journal of Pharmacology and Experimental Therapeutics","topic":"Cannabis and Cannabinoid Research","field":"Medicine","cited_by":61,"is_retracted":false,"has_abstract":false,"ca_institutions":"University of Calgary","funders":"Canadian Institutes of Health Research","keywords":"AM251; Cannabinoid receptor type 2; Cannabinoid receptor; Cannabinoid; Pharmacology; Chemistry; Agonist; Receptor; Cannabinoid receptor antagonist; Motility; Colitis; Receptor antagonist; Knockout mouse; Cannabinoid Receptor Agonists; Internal medicine; Endocrinology; Antagonist; Biochemistry; Medicine; Biology; Cell biology","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.00007845188,0.0002883515,0.0003382553,0.0002581107,0.0001517254,0.000114528,0.0002900488,0.0002249751,0.003607339],"category_scores_gemma":[0.0001018947,0.0001433773,0.0002174291,0.0001408797,0.000234149,0.000189527,0.0001889008,0.0006024581,0.0009807363],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0001785573,"about_ca_system_score_gemma":0.0004035668,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.001355567,"about_ca_topic_score_gemma":0.003789695,"domain_scores_codex":[0.9999112,0.000009640434,0.000005000971,0.00001024278,0.00002115547,0.00004286649],"domain_scores_gemma":[0.9999344,0.000008207827,0.0000154186,0.000007706576,0.000005732244,0.00002849984],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.00114814,0.0001236747,0.0001715897,0.00009054732,0.00001311493,0.0001737442,0.00001673204,0.000131403,0.9914604,0.0001431594,0.0002025302,0.00632497],"study_design_scores_gemma":[0.0003076372,0.003655529,0.004594992,0.00002106366,0.00003775637,0.0006227869,0.0000618981,0.0009400116,0.9859025,0.0001254987,0.003715436,0.00001481655],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9897584,0.002144489,0.001638089,0.0002272818,0.0001193441,0.00004430746,0.000607677,0.0001807818,0.005279727],"genre_scores_gemma":[0.9913855,0.001581825,0.00131689,0.00009115527,0.00002000942,0.00003588885,0.0005887057,0.00001596783,0.00496408],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.003607339,"threshold_uncertainty_score":0.01206774,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.02274606643272663,"score_gpt":0.3379344917067155,"score_spread":0.3151884252739889,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}