{"id":"W2114763268","doi":"10.1017/s1462399411001992","title":"Bromodomains as therapeutic targets","year":2011,"lang":"en","type":"review","venue":"Expert Reviews in Molecular Medicine","topic":"Peptidase Inhibition and Analysis","field":"Medicine","cited_by":436,"is_retracted":false,"has_abstract":true,"ca_institutions":"","funders":"Knut och Alice Wallenbergs Stiftelse; Karolinska Institutet; Stiftelsen för Strategisk Forskning; Ontario Genomics Institute; Canadian Institutes of Health Research; Ontario Genomics; Genome Canada; Ontario Innovation Trust; Wellcome Trust; GlaxoSmithKline","keywords":"Bromodomain; Acetylation; Lysine; Histone Acetyltransferases; Histone; BRD4; Drug development; Computational biology; Epigenetics; Biochemistry; Biology; Chemistry; Small molecule; Drug discovery; Cell biology; Amino acid; Drug; Pharmacology; Gene","routes":{"ca_aff":false,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":true},"retraction":null,"screen":null,"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.08277281613059019,"score_gpt":0.4057593280628275,"score_spread":0.3229865119322373,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}