{"id":"W2126816965","doi":"10.2174/15672018113109990038","title":"Pharmacokinetics of 3&amp;#8217;-O-Retinoyl-5-fluoro-2&amp;#8217;-deoxyuridine (RFUdR), a Dual Acting Mutually Masking Prodrug, and Its Metabolites in Tumor Bearing Mice","year":2013,"lang":"en","type":"article","venue":"Current Drug Delivery","topic":"Retinoids in leukemia and cellular processes","field":"Biochemistry, Genetics and Molecular Biology","cited_by":2,"is_retracted":false,"has_abstract":true,"ca_institutions":"Alberta Energy","funders":"Canadian Institutes of Health Research","keywords":"Prodrug; Pharmacokinetics; Deoxyuridine; Chemistry; Bolus (digestion); Metabolite; Pharmacology; Bioavailability; Retinoic acid; Oral administration; High-performance liquid chromatography; Active metabolite; Medicine; Internal medicine; Biochemistry; Chromatography","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0001923982,0.0002806492,0.0003728884,0.000213214,0.00008239393,0.0003436125,0.0001557507,0.0003157125,0.0005289299],"category_scores_gemma":[0.000269959,0.0002643734,0.0002439349,0.0001542974,0.0002816769,0.0003259236,0.00007849326,0.0006356979,0.0003900297],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.000388793,"about_ca_system_score_gemma":0.0002978741,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.001094231,"about_ca_topic_score_gemma":0.0007698598,"domain_scores_codex":[0.9999027,0.00002398444,0.000003486845,0.00002700191,0.00001610936,0.00002674698],"domain_scores_gemma":[0.9998724,0.00003297808,0.00003919128,0.00001575345,0.00001167393,0.00002793021],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.006701787,0.0002127497,0.001924151,0.00005946583,0.00003384079,0.0001033038,0.0001186793,0.00137247,0.9706343,0.0003034367,0.0003297238,0.01820598],"study_design_scores_gemma":[0.0002960416,0.01340975,0.01661506,0.00001585489,0.0001191975,0.0005140138,0.00007824432,0.009976165,0.9531898,0.0002502429,0.005497312,0.00003832811],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9926155,0.00208419,0.003251111,0.0000746807,0.00001887392,0.0000298705,0.0005836322,0.0001669688,0.001175238],"genre_scores_gemma":[0.9933085,0.001088323,0.002004315,0.00005474125,0.00001461106,0.00006399143,0.0006085018,0.00004624311,0.002810685],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.001094231,"threshold_uncertainty_score":0.002820849,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.0188955237968077,"score_gpt":0.2696374619946643,"score_spread":0.2507419381978566,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}