{"id":"W2156373035","doi":"10.1021/cb500129t","title":"Exploration of Type II Binding Mode: A Privileged Approach for Kinase Inhibitor Focused Drug Discovery?","year":2014,"lang":"en","type":"review","venue":"ACS Chemical Biology","topic":"HER2/EGFR in Cancer Research","field":"Medicine","cited_by":428,"is_retracted":false,"has_abstract":true,"ca_institutions":"","funders":"Canadian Institutes of Health Research; Wellcome Trust","keywords":"Small molecule; Drug discovery; Kinase; Binding site; Chemistry; Stereochemistry; Active site; Plasma protein binding; Biophysics; Enzyme; Combinatorial chemistry; Biochemistry; Biology","routes":{"ca_aff":false,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":true},"retraction":null,"screen":null,"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.1308690158421731,"score_gpt":0.4185566617117618,"score_spread":0.2876876458695887,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}