{"id":"W2159467223","doi":"10.1124/dmd.108.023101","title":"Deferiprone Glucuronidation by Human Tissues and Recombinant UDP Glucuronosyltransferase 1A6: An in Vitro Investigation of Genetic and Splice Variants","year":2008,"lang":"en","type":"article","venue":"Drug Metabolism and Disposition","topic":"Neonatal Health and Biochemistry","field":"Medicine","cited_by":51,"is_retracted":false,"has_abstract":false,"ca_institutions":"Université Laval; Centre hospitalier universitaire de Québec","funders":"","keywords":"Deferiprone; Glucuronidation; Microsome; UGT2B7; Metabolite; Pharmacology; Chemistry; Glucuronosyltransferase; In vitro; Biochemistry; Isozyme; Deferoxamine; Biology; Enzyme","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"codex-gemma-dda1882f352a","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0001283189,0.0001250632,0.0002389982,0.00006936255,0.0001044152,0.000008217589,0.00002286385,0.00007416382,0.000005417336],"category_scores_gemma":[0.000008564721,0.0001175232,0.0000126172,0.0001048128,0.0001295803,0.0001855826,0.00001223506,0.00008875223,4.177838e-7],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.00001117743,"about_ca_system_score_gemma":0.00002896987,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0005674983,"about_ca_topic_score_gemma":0.00001602062,"domain_scores_codex":[0.9991378,0.00005644913,0.0002720505,0.0002683931,0.0001189518,0.0001464003],"domain_scores_gemma":[0.9995742,0.00001458315,0.00006362097,0.0001104064,0.00003557279,0.0002016262],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"observational","study_design_scores_codex":[0.0003623521,0.0001162011,0.01111752,0.0003860656,0.000005675126,0.00001014377,0.001084753,9.878451e-8,0.9721152,0.00007054873,0.00002730937,0.01470417],"study_design_scores_gemma":[0.001955455,0.0001156507,0.5700713,0.00007454861,0.00006382649,0.00009406771,0.0001271331,0.00008844244,0.4269484,0.00025013,0.00009182285,0.0001191703],"study_design_candidate":"bench_or_experimental","study_design_consensus":null,"genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9906058,0.008718173,0.00005537243,0.0001988356,0.00003363398,0.000298659,0.00004903827,0.00001429013,0.00002621638],"genre_scores_gemma":[0.9955517,0.002907681,0.0006905562,0.0001319566,0.00004698396,0.00001561468,0.0006163952,0.00001051849,0.00002860493],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.5589538,"threshold_uncertainty_score":0.4792458,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.009921851346929833,"score_gpt":0.2496478314606932,"score_spread":0.2397259801137633,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}