{"id":"W2159467223","doi":"10.1124/dmd.108.023101","title":"Deferiprone Glucuronidation by Human Tissues and Recombinant UDP Glucuronosyltransferase 1A6: An in Vitro Investigation of Genetic and Splice Variants","year":2008,"lang":"en","type":"article","venue":"Drug Metabolism and Disposition","topic":"Neonatal Health and Biochemistry","field":"Medicine","cited_by":51,"is_retracted":false,"has_abstract":false,"ca_institutions":"Université Laval; Centre hospitalier universitaire de Québec","funders":"","keywords":"Deferiprone; Glucuronidation; Microsome; UGT2B7; Metabolite; Pharmacology; Chemistry; Glucuronosyltransferase; In vitro; Biochemistry; Isozyme; Deferoxamine; Biology; Enzyme","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0004777272,0.0004717206,0.0003759671,0.0002495167,0.0002114053,0.0004101373,0.0002745732,0.0002226264,0.001140461],"category_scores_gemma":[0.0004686901,0.0002854746,0.0004423294,0.0003597589,0.0002443749,0.0002334717,0.0001616224,0.0005101548,0.0004743928],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0003575708,"about_ca_system_score_gemma":0.0002553439,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.002867284,"about_ca_topic_score_gemma":0.002096461,"domain_scores_codex":[0.9996775,0.0001493492,0.00003055171,0.00006048703,0.00003946746,0.0000427316],"domain_scores_gemma":[0.9997756,0.0000954289,0.00002789519,0.00004626335,0.00003199881,0.00002285912],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.002147757,0.00009824409,0.001200545,0.00007960435,0.00004794861,0.0001868211,0.0001145517,0.0003328027,0.9920141,0.0003286043,0.0001054325,0.003343598],"study_design_scores_gemma":[0.00006169167,0.0007861212,0.003709927,0.000009184317,0.00009317821,0.001122661,0.00006642162,0.001890948,0.9899625,0.0000851873,0.00219997,0.00001208516],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9898419,0.003746391,0.004591516,0.00007843476,0.00003614413,0.0000238618,0.000598699,0.00003784438,0.001045298],"genre_scores_gemma":[0.9888072,0.001671939,0.004212469,0.00003604539,0.00002180252,0.00001784646,0.003145879,0.00004472853,0.002042038],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.002867284,"threshold_uncertainty_score":0.005701184,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.009921851346929833,"score_gpt":0.2496478314606932,"score_spread":0.2397259801137633,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}