{"id":"W2165528419","doi":"10.1139/y02-041","title":"Biochemical and pharmacological activities of SSR 146977, a new potent nonpeptide tachykinin NK<sub>3</sub> receptor antagonist","year":2002,"lang":"en","type":"article","venue":"Canadian Journal of Physiology and Pharmacology","topic":"Neuropeptides and Animal Physiology","field":"Neuroscience","cited_by":38,"is_retracted":false,"has_abstract":true,"ca_institutions":"","funders":"","keywords":"Endocrinology; Internal medicine; Neurokinin B; Tachykinin receptor; Neurokinin A; Chemistry; Receptor antagonist; Acetylcholine; Receptor; Biology; Pharmacology; Substance P; Antagonist; Neuropeptide; Medicine","routes":{"ca_aff":false,"ca_fund":false,"ca_venue":true,"about_ca":false,"invisible_to_affiliation_only":true},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0001514462,0.0004478012,0.0006521104,0.0002766897,0.0001419489,0.0002522495,0.0003246416,0.0003161306,0.001666319],"category_scores_gemma":[0.0001426906,0.0002297421,0.0004269398,0.0002309718,0.0001857099,0.000231869,0.0001625015,0.0006584646,0.001103599],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0001983082,"about_ca_system_score_gemma":0.0002848325,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.000450278,"about_ca_topic_score_gemma":0.0007879223,"domain_scores_codex":[0.9998776,0.00002427682,0.00002036992,0.00001471891,0.00003181277,0.00003115274],"domain_scores_gemma":[0.999938,0.000008518402,0.00001462717,0.000007213675,0.00001355342,0.00001795842],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0007394931,0.0001222525,0.0002983317,0.0001662835,0.00003719575,0.0002447374,0.00001840266,0.00020553,0.9874849,0.0001682981,0.0002430179,0.0102716],"study_design_scores_gemma":[0.0004014939,0.004897632,0.01454877,0.00002248169,0.0002293559,0.004050257,0.00003745014,0.002204372,0.9606623,0.0001436704,0.01276334,0.00003883488],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9598481,0.02284477,0.005991877,0.0002921872,0.00008544948,0.0001592134,0.001583332,0.0002354728,0.008959519],"genre_scores_gemma":[0.9631105,0.01761037,0.007208622,0.0002912696,0.00008755865,0.0001915881,0.006144128,0.00005021937,0.005305722],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.001666319,"threshold_uncertainty_score":0.005574346,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.03108501279926275,"score_gpt":0.2577718028641278,"score_spread":0.2266867900648651,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}