{"id":"W2166163013","doi":"10.18433/j3501w","title":"Transport Characteristics of Tryptanthrin and its Inhibitory Effect on P-gp and MRP2 in Caco-2 Cells","year":2011,"lang":"en","type":"article","venue":"Journal of Pharmacy & Pharmaceutical Sciences","topic":"Quinazolinone synthesis and applications","field":"Chemistry","cited_by":38,"is_retracted":false,"has_abstract":true,"ca_institutions":"","funders":"Northwest University","keywords":"Caco-2; Multidrug resistance-associated protein 2; Chemistry; Inhibitory postsynaptic potential; Pharmacology; Traditional medicine; Biochemistry; Transporter; In vitro; Biology; Medicine; ATP-binding cassette transporter; Endocrinology; Gene","routes":{"ca_aff":false,"ca_fund":false,"ca_venue":true,"about_ca":false,"invisible_to_affiliation_only":true},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0001906619,0.0002379618,0.0003302377,0.0001905132,0.0001852266,0.0002527474,0.0001071636,0.0002594161,0.001030774],"category_scores_gemma":[0.0001679768,0.0001215273,0.0003532198,0.0003499243,0.0001520949,0.0003435542,0.0000844065,0.000367608,0.0002748294],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0002388533,"about_ca_system_score_gemma":0.000134824,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.001460049,"about_ca_topic_score_gemma":0.001063016,"domain_scores_codex":[0.9998133,0.00004126487,0.00002200004,0.00003127295,0.00006452348,0.0000277284],"domain_scores_gemma":[0.9999015,0.00003029786,0.00001922258,0.00001188749,0.00002604044,0.00001103813],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0002279906,0.00003706471,0.0003443925,0.0001058285,0.000008803801,0.0001732178,0.00003782637,0.0000855101,0.9974994,0.00004975645,0.00007688694,0.001353322],"study_design_scores_gemma":[0.00004990639,0.001228837,0.02504322,0.00001383399,0.00007583647,0.001557869,0.0001087103,0.003274425,0.9633573,0.00004829754,0.005224193,0.00001751615],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9867905,0.007245989,0.002329878,0.000338469,0.00004178269,0.00003999057,0.0009296938,0.00007672681,0.002207046],"genre_scores_gemma":[0.98998,0.003296573,0.002817371,0.00008404438,0.00002746061,0.00004940153,0.001002247,0.00001243061,0.002730354],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.001460049,"threshold_uncertainty_score":0.003448308,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.06231012022621672,"score_gpt":0.3465562825463321,"score_spread":0.2842461623201154,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}