{"id":"W2325404207","doi":"10.1158/1538-7445.am2013-1070","title":"Abstract 1070: New potent inhibitors of the androgen receptor that target its BF3 surface binding site.","year":2013,"lang":"en","type":"article","venue":"Cancer Research","topic":"Prostate Cancer Treatment and Research","field":"Medicine","cited_by":1,"is_retracted":false,"has_abstract":true,"ca_institutions":"","funders":"","keywords":"Transactivation; Androgen receptor; Bicalutamide; Prostate cancer; LNCaP; Antiandrogens; Chemistry; Cancer research; Binding site; In silico; Dihydrotestosterone; Pharmacology; Cancer; Androgen; Biochemistry; Biology; Internal medicine; Medicine; Transcription factor; Hormone","routes":{"ca_aff":false,"ca_fund":false,"ca_venue":false,"about_ca":true,"invisible_to_affiliation_only":true},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0001096945,0.0006856198,0.0003639534,0.00038248,0.0001376544,0.0002375277,0.0004607091,0.000313093,0.002200805],"category_scores_gemma":[0.0001085019,0.0001335133,0.0003445385,0.0004012499,0.0001828683,0.0001440105,0.0001888104,0.0005262576,0.001295771],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0004329057,"about_ca_system_score_gemma":0.0003602397,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.002334023,"about_ca_topic_score_gemma":0.003940974,"domain_scores_codex":[0.9999342,0.000009880972,0.00000334976,0.00001030347,0.00002646397,0.00001586198],"domain_scores_gemma":[0.9999702,0.000006014939,0.000007227942,0.000001798679,0.000003574844,0.00001111823],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.001073404,0.0005282169,0.001157266,0.0005754617,0.00007735132,0.0004983156,0.00004445155,0.005565497,0.8980798,0.001920684,0.005234043,0.08524548],"study_design_scores_gemma":[0.001522846,0.006343929,0.01022251,0.0001391526,0.0002303791,0.00286962,0.00005790246,0.01810003,0.8793704,0.001283975,0.07975266,0.0001065058],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.8744785,0.04346738,0.03513128,0.000810683,0.0003177617,0.0007185823,0.008735164,0.002152563,0.03418818],"genre_scores_gemma":[0.9342276,0.01576155,0.02174138,0.0006785862,0.00003448647,0.0002898976,0.009763057,0.0001271986,0.01737629],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.002334023,"threshold_uncertainty_score":0.007362425,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.1040328123437652,"score_gpt":0.3842405442031027,"score_spread":0.2802077318593375,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}