{"id":"W2427814062","doi":"10.1021/acs.molpharmaceut.5b00070","title":"Imaging Bradykinin B1 Receptor with<sup>68</sup>Ga-Labeled [des-Arg<sup>10</sup>]Kallidin Derivatives: Effect of the Linker on Biodistribution and Tumor Uptake","year":2015,"lang":"en","type":"article","venue":"Molecular Pharmaceutics","topic":"Coagulation, Bradykinin, Polyphosphates, and Angioedema","field":"Medicine","cited_by":23,"is_retracted":false,"has_abstract":true,"ca_institutions":"University of British Columbia; BC Cancer Agency","funders":"Canadian Institutes of Health Research; Leading Edge Endowment Fund","keywords":"Biodistribution; Linker; HEK 293 cells; Chemistry; Receptor; In vivo; Pharmacokinetics; Bradykinin; Molecular biology; In vitro; Cancer research; Biochemistry; Pharmacology; Medicine; Biology","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0002236826,0.0003429835,0.0002638864,0.00008581192,0.00006667671,0.0002190555,0.0002379221,0.0003339467,0.0004487025],"category_scores_gemma":[0.0001813584,0.0001694663,0.0001289669,0.0001082796,0.0001438629,0.0002677992,0.0001178289,0.0003145822,0.0001994165],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0003240745,"about_ca_system_score_gemma":0.0001621965,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0004909896,"about_ca_topic_score_gemma":0.0005427253,"domain_scores_codex":[0.999907,0.00002529462,0.000005520312,0.00002198893,0.00001972865,0.00002044849],"domain_scores_gemma":[0.9998958,0.00003105749,0.00003882335,0.000005855744,0.00001071278,0.00001768411],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0001244771,0.000009352263,0.00006906539,0.00002467365,0.000003273789,0.00001564667,0.000007546728,0.00008498891,0.998882,0.00001424267,0.000009567273,0.0007552564],"study_design_scores_gemma":[0.00001711822,0.0004011838,0.0009951908,0.000002096781,0.000016163,0.0002027484,0.000009512007,0.001108149,0.9967687,0.00000804216,0.0004666499,0.000004358828],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9957572,0.001145052,0.002590801,0.00003589333,0.000005357532,0.00001478974,0.00005325584,0.00002961032,0.0003680549],"genre_scores_gemma":[0.9832544,0.001491839,0.01360759,0.00008085475,0.000007698123,0.00004429119,0.000262836,0.00003576031,0.001214811],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.0004909896,"threshold_uncertainty_score":0.002351284,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.02811547747883363,"score_gpt":0.2990557724212209,"score_spread":0.2709402949423872,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}