{"id":"W2427814062","doi":"10.1021/acs.molpharmaceut.5b00070","title":"Imaging Bradykinin B1 Receptor with<sup>68</sup>Ga-Labeled [des-Arg<sup>10</sup>]Kallidin Derivatives: Effect of the Linker on Biodistribution and Tumor Uptake","year":2015,"lang":"en","type":"article","venue":"Molecular Pharmaceutics","topic":"Coagulation, Bradykinin, Polyphosphates, and Angioedema","field":"Medicine","cited_by":23,"is_retracted":false,"has_abstract":true,"ca_institutions":"University of British Columbia; BC Cancer Agency","funders":"Canadian Institutes of Health Research; Leading Edge Endowment Fund","keywords":"Biodistribution; Linker; HEK 293 cells; Chemistry; Receptor; In vivo; Pharmacokinetics; Bradykinin; Molecular biology; In vitro; Cancer research; Biochemistry; Pharmacology; Medicine; Biology","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"codex-gemma-dda1882f352a","candidate_categories":["metaepi_narrow"],"consensus_categories":[],"category_scores_codex":[0.0008554006,0.0005363332,0.0006607948,0.0001534406,0.0002212283,0.00006976026,0.0002473751,0.000128521,0.0001347468],"category_scores_gemma":[0.000561281,0.0003854319,0.0002163053,0.000671283,0.0005146977,0.000159049,0.0001339022,0.0004523474,0.00005253666],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.000212791,"about_ca_system_score_gemma":0.0002464025,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.00003159452,"about_ca_topic_score_gemma":0.000001103003,"domain_scores_codex":[0.997021,0.0004165065,0.0005962714,0.0005901451,0.0007777454,0.0005983448],"domain_scores_gemma":[0.9981089,0.0002171219,0.000295787,0.0005740834,0.000371409,0.0004327451],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"observational","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.01219341,0.002364721,0.4340823,0.002762256,0.002813601,0.0008017033,0.01296643,0.01218146,0.4051583,0.001607297,0.02009235,0.0929761],"study_design_scores_gemma":[0.01532376,0.001610594,0.007959252,0.001114981,0.001210523,0.0002513834,0.0004994185,0.06630429,0.8433353,0.00011436,0.06146961,0.0008065275],"study_design_candidate":"bench_or_experimental","study_design_consensus":null,"genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9912844,0.004811882,0.0007712342,0.001204893,0.0001089207,0.001184967,0.0001019671,0.0001242617,0.0004075007],"genre_scores_gemma":[0.9971956,0.0001426813,0.0007683247,0.001106328,0.0001455568,0.00004636692,0.0001934224,0.00008965946,0.0003120553],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.438177,"threshold_uncertainty_score":0.9998598,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.02811547747883363,"score_gpt":0.2990557724212209,"score_spread":0.2709402949423872,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}