{"id":"W2550163245","doi":"10.1016/j.bmc.2016.11.038","title":"Synthesis and evaluation of a 68Ga-labeled bradykinin B1 receptor agonist for imaging with positron emission tomography","year":2016,"lang":"en","type":"article","venue":"Bioorganic & Medicinal Chemistry","topic":"Peptidase Inhibition and Analysis","field":"Medicine","cited_by":4,"is_retracted":false,"has_abstract":false,"ca_institutions":"University of British Columbia; BC Cancer Agency","funders":"Canadian Institutes of Health Research","keywords":"Chemistry; Biodistribution; Positron emission tomography; In vivo; Agonist; Bradykinin; Clearance; Receptor; In vitro; Pet imaging; Nuclear medicine; Biochemistry; Medicine","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0002489577,0.000401624,0.0003422657,0.0002485873,0.0003434817,0.0003503947,0.0005222629,0.0004792095,0.001131518],"category_scores_gemma":[0.0001907986,0.0002490066,0.0002683004,0.0002505532,0.0001646616,0.0002885112,0.0002165482,0.0004831145,0.0007771386],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0003945216,"about_ca_system_score_gemma":0.0005884307,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.001888582,"about_ca_topic_score_gemma":0.002244825,"domain_scores_codex":[0.9998664,0.00002639171,0.000008360438,0.00002293846,0.00003051997,0.00004546309],"domain_scores_gemma":[0.9999279,0.000007809707,0.00001143648,0.000008200981,0.00002009621,0.00002448835],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0002645335,0.0001830637,0.000124341,0.000148434,0.00002724809,0.0005292313,0.00007539945,0.001342482,0.9856629,0.0007243502,0.0003420482,0.010576],"study_design_scores_gemma":[0.00007684306,0.001261424,0.0006051471,0.00001400992,0.00006364131,0.0007055892,0.00003520786,0.001496776,0.9790893,0.00009493087,0.0165289,0.00002830689],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.908379,0.009529657,0.06025193,0.0007044418,0.0001655915,0.000863147,0.001395465,0.0002915908,0.01841937],"genre_scores_gemma":[0.9602301,0.004941899,0.02358698,0.0002095767,0.00003482036,0.0001314182,0.001392663,0.00006943545,0.009403194],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.001888582,"threshold_uncertainty_score":0.003785253,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.01388681263952685,"score_gpt":0.2675048122196557,"score_spread":0.2536179995801289,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}