{"id":"W2550163245","doi":"10.1016/j.bmc.2016.11.038","title":"Synthesis and evaluation of a 68Ga-labeled bradykinin B1 receptor agonist for imaging with positron emission tomography","year":2016,"lang":"en","type":"article","venue":"Bioorganic & Medicinal Chemistry","topic":"Peptidase Inhibition and Analysis","field":"Medicine","cited_by":4,"is_retracted":false,"has_abstract":false,"ca_institutions":"University of British Columbia; BC Cancer Agency","funders":"Canadian Institutes of Health Research","keywords":"Chemistry; Biodistribution; Positron emission tomography; In vivo; Agonist; Bradykinin; Clearance; Receptor; In vitro; Pet imaging; Nuclear medicine; Biochemistry; Medicine","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"codex-gemma-dda1882f352a","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0005900432,0.0001819718,0.0003528661,0.00008043509,0.00007603435,0.000009006051,0.00006449005,0.00006691807,0.000745155],"category_scores_gemma":[0.0005209984,0.0001115909,0.00009467154,0.0002424962,0.0002053167,0.00005614271,0.00001927047,0.00007831887,0.000002158404],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.000105798,"about_ca_system_score_gemma":0.0002245617,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.00001039376,"about_ca_topic_score_gemma":0.000001021597,"domain_scores_codex":[0.9985203,0.00003510258,0.000310288,0.0003438226,0.0005827362,0.0002077398],"domain_scores_gemma":[0.998805,0.0001599767,0.0001992424,0.0002434728,0.0003774525,0.0002148299],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0003458492,0.000098099,0.00621371,0.0002599678,0.0001102104,0.000004197189,0.00004410988,1.35024e-8,0.9783733,0.000002759077,0.00109208,0.01345565],"study_design_scores_gemma":[0.003418654,0.0001146572,0.002110152,0.003215797,0.0009672595,0.0001160065,0.0002883962,0.0001305378,0.9891164,0.00002464259,0.0003475891,0.0001499156],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9939861,0.0006290684,0.000343685,0.004145031,0.00001369495,0.0002512832,0.00004239066,0.00004439963,0.0005443541],"genre_scores_gemma":[0.9987819,0.00004346444,0.000437532,0.0001237147,0.0001820797,0.00004290498,0.00004722805,0.0000250226,0.0003161888],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.01330573,"threshold_uncertainty_score":0.8158925,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.01388681263952685,"score_gpt":0.2675048122196557,"score_spread":0.2536179995801289,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}