{"id":"W2561387856","doi":"10.1158/1538-7445.am2015-3652","title":"Abstract 3652: Development of novel chemical inhibitors targeting the N-terminal domain (NTD) of androgen receptor variants as anti-prostate cancer agents","year":2015,"lang":"en","type":"article","venue":"Cancer Research","topic":"Prostate Cancer Treatment and Research","field":"Medicine","cited_by":0,"is_retracted":false,"has_abstract":true,"ca_institutions":"McGill University","funders":"","keywords":"Enzalutamide; Bicalutamide; Prostate cancer; Androgen receptor; Cancer research; Antiandrogens; Medicine; Cancer; Androgen; Androgen deprivation therapy; Internal medicine; Hormone","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0001103938,0.0004692987,0.0003533554,0.0002700087,0.000114157,0.0002607733,0.0003697863,0.0002844767,0.0022808],"category_scores_gemma":[0.00004809627,0.0001288477,0.0003485725,0.0001911276,0.0001129993,0.0001843246,0.000165202,0.0005556875,0.0007290696],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0002457926,"about_ca_system_score_gemma":0.0003163413,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0008675907,"about_ca_topic_score_gemma":0.001232593,"domain_scores_codex":[0.9999475,0.000005939854,0.000004207732,0.00001123322,0.00001638474,0.00001473216],"domain_scores_gemma":[0.9999793,9.866554e-7,0.000003779547,0.000001191022,0.000004365722,0.00001038376],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.000897624,0.0007566321,0.0005756228,0.000650139,0.0001157615,0.0004187461,0.00003361164,0.001614775,0.9314345,0.002144597,0.003293397,0.05806449],"study_design_scores_gemma":[0.001928196,0.01247893,0.008558654,0.0001405353,0.0003876849,0.002690241,0.00004982445,0.007161499,0.7967774,0.0007854592,0.1689541,0.00008742612],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.873616,0.06620073,0.02122955,0.001034746,0.001114055,0.0009489859,0.003654235,0.000678037,0.03152366],"genre_scores_gemma":[0.9420025,0.02306958,0.01030282,0.0007708736,0.00008156146,0.0003449894,0.003728644,0.00004851473,0.01965055],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.0022808,"threshold_uncertainty_score":0.00763005,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.120834366788184,"score_gpt":0.4247683232650827,"score_spread":0.3039339564768987,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}