{"id":"W2571708387","doi":"10.1021/acs.molpharmaceut.6b01055","title":"Radiolabeled R954 Derivatives for Imaging Bradykinin B1 Receptor Expression with Positron Emission Tomography","year":2017,"lang":"en","type":"article","venue":"Molecular Pharmaceutics","topic":"Coagulation, Bradykinin, Polyphosphates, and Angioedema","field":"Medicine","cited_by":8,"is_retracted":false,"has_abstract":true,"ca_institutions":"University of British Columbia; BC Cancer Agency","funders":"Institute of Cancer Research; Canadian Institutes of Health Research; Leading Edge Endowment Fund","keywords":"Positron emission tomography; Positron Emission Tomography-Computed Tomography; Brain positron emission tomography; Bradykinin; Nuclear medicine; Chemistry; Pet imaging; Receptor; Medicine; Preclinical imaging; Biochemistry; Biology; In vivo; Genetics","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0004183831,0.0005497414,0.0003605291,0.0002579408,0.00009616777,0.0003439629,0.0005612238,0.0007006493,0.002262168],"category_scores_gemma":[0.0002211558,0.0003935628,0.0002297153,0.0003308002,0.0001626953,0.0003552667,0.0002457007,0.0006238516,0.0008528755],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0004855519,"about_ca_system_score_gemma":0.0001826308,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0008518262,"about_ca_topic_score_gemma":0.001444432,"domain_scores_codex":[0.9997682,0.00008114657,0.00001200133,0.00004575805,0.00004088712,0.00005198524],"domain_scores_gemma":[0.9999306,0.00002128798,0.00001711578,0.000008006132,0.00001084356,0.00001212036],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0001691358,0.00002902828,0.00008657423,0.0000949594,0.00001181539,0.00007809061,0.00001875516,0.0003026646,0.9962088,0.0002300167,0.0001786343,0.002591613],"study_design_scores_gemma":[0.00007091778,0.0006475879,0.0008993881,0.00001509059,0.00003663914,0.0006074099,0.00002454296,0.003088325,0.9861466,0.00007547438,0.008360405,0.00002760897],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.8917494,0.01876059,0.07751139,0.0004457717,0.00009502575,0.0003656895,0.001171509,0.000500814,0.009399806],"genre_scores_gemma":[0.885152,0.009552117,0.0938122,0.0002919206,0.00002815727,0.0003603556,0.001861604,0.0001717064,0.008769814],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.002262168,"threshold_uncertainty_score":0.007567704,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.02316130767556829,"score_gpt":0.332332839995903,"score_spread":0.3091715323203347,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}