{"id":"W2571708387","doi":"10.1021/acs.molpharmaceut.6b01055","title":"Radiolabeled R954 Derivatives for Imaging Bradykinin B1 Receptor Expression with Positron Emission Tomography","year":2017,"lang":"en","type":"article","venue":"Molecular Pharmaceutics","topic":"Coagulation, Bradykinin, Polyphosphates, and Angioedema","field":"Medicine","cited_by":8,"is_retracted":false,"has_abstract":true,"ca_institutions":"University of British Columbia; BC Cancer Agency","funders":"Institute of Cancer Research; Canadian Institutes of Health Research; Leading Edge Endowment Fund","keywords":"Positron emission tomography; Positron Emission Tomography-Computed Tomography; Brain positron emission tomography; Bradykinin; Nuclear medicine; Chemistry; Pet imaging; Receptor; Medicine; Preclinical imaging; Biochemistry; Biology; In vivo; Genetics","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"codex-gemma-dda1882f352a","candidate_categories":["metaepi_narrow"],"consensus_categories":[],"category_scores_codex":[0.0002265731,0.0003406826,0.0003983568,0.0001480013,0.0006645739,0.0001464971,0.0002762364,0.00009803745,0.00005916307],"category_scores_gemma":[0.0001278137,0.0002822778,0.0002178999,0.0001245428,0.0001885979,0.00026531,0.00009422674,0.0002136539,0.000005046428],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.00005445039,"about_ca_system_score_gemma":0.0001017902,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.00001548043,"about_ca_topic_score_gemma":8.989946e-7,"domain_scores_codex":[0.9982598,0.00006235886,0.0003197421,0.0004960327,0.0003784778,0.0004836145],"domain_scores_gemma":[0.9984144,0.0000734352,0.0003142784,0.000663125,0.0002099385,0.0003248464],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0008031889,0.0001635766,0.1024453,0.0001416621,0.0001423491,0.00004727376,0.0003461625,0.00001054746,0.8754278,0.0001049292,0.001886165,0.01848105],"study_design_scores_gemma":[0.005610513,0.0002142754,0.00985526,0.0005156704,0.0003069659,0.00004342063,0.00008526606,0.003915954,0.9498171,0.0001210896,0.02912965,0.0003848661],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9666125,0.005060425,0.02258241,0.002897088,0.0003830424,0.00131135,0.00003129048,0.0001964913,0.0009254367],"genre_scores_gemma":[0.9854815,0.0001553123,0.01231997,0.000934392,0.0002835417,0.00006521076,0.0001316337,0.00009505994,0.0005333844],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.09259003,"threshold_uncertainty_score":0.9999629,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.02316130767556829,"score_gpt":0.332332839995903,"score_spread":0.3091715323203347,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}