{"id":"W2573175803","doi":"10.7717/peerj.2911","title":"Species-specific pharmacology of maximakinin, an amphibian homologue of bradykinin: putative prodrug activity at the human B <sub>2</sub> receptor and peptidase resistance in rats","year":2017,"lang":"en","type":"article","venue":"PeerJ","topic":"Coagulation, Bradykinin, Polyphosphates, and Angioedema","field":"Medicine","cited_by":7,"is_retracted":false,"has_abstract":true,"ca_institutions":"Université Laval","funders":"Canadian Institutes of Health Research","keywords":"Bradykinin; Receptor; Molecular biology; Histamine; Agonist; Recombinant DNA; Peptide; Chemistry; Radioligand; Biology; Biochemistry; Pharmacology","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"codex-gemma-dda1882f352a","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0006150491,0.0002450021,0.0006320394,0.0001366278,0.0003827787,0.00003021954,0.000260789,0.0001219421,0.0001634565],"category_scores_gemma":[0.0001487352,0.0001990419,0.0001116482,0.0001421628,0.001148869,0.0002608654,0.000153756,0.0002407602,0.000007570174],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0001085554,"about_ca_system_score_gemma":0.00009724993,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0001399877,"about_ca_topic_score_gemma":0.001865978,"domain_scores_codex":[0.9982135,0.0001947202,0.0004511812,0.0004941054,0.0003142424,0.0003322414],"domain_scores_gemma":[0.9981593,0.0002134672,0.0006308286,0.0006667859,0.000199527,0.0001300592],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"observational","study_design_scores_codex":[0.001064448,0.0004257249,0.08963161,0.0001575393,0.00007694388,0.00005677019,0.004852231,0.00000297052,0.8920075,0.0007223807,0.005419732,0.005582168],"study_design_scores_gemma":[0.001490326,0.0001800686,0.5468255,0.00008079805,0.0000390619,0.000009796446,0.0001495936,0.00001596235,0.4493391,0.0002131781,0.001535978,0.0001205758],"study_design_candidate":"bench_or_experimental","study_design_consensus":null,"genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9941276,0.0009217327,0.000007181529,0.002437967,0.0002319264,0.0006818816,0.0001140299,0.00002630188,0.001451326],"genre_scores_gemma":[0.9975706,0.0001751241,0.000133825,0.0000828484,0.000240543,0.00003451193,0.00006160875,0.00003178148,0.001669126],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.4571939,"threshold_uncertainty_score":0.8116695,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.03903488813849881,"score_gpt":0.313152889135241,"score_spread":0.2741180009967422,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}