{"id":"W2770571637","doi":"10.1016/j.nucmedbio.2017.11.004","title":"Synthesis, in vitro and in vivo evaluation of 18F-fluoronorimatinib as radiotracer for Imatinib-sensitive gastrointestinal stromal tumors","year":2017,"lang":"en","type":"article","venue":"Nuclear Medicine and Biology","topic":"Gastrointestinal Tumor Research and Treatment","field":"Medicine","cited_by":4,"is_retracted":false,"has_abstract":false,"ca_institutions":"University of Alberta","funders":"Deutsche Forschungsgemeinschaft","keywords":"GiST; Imatinib; Radioligand; In vivo; Stromal tumor; Cancer research; Tyrosine-kinase inhibitor; Stromal cell; Chemistry; Positron emission tomography; In vitro; Biodistribution; Medicine; Pharmacology; Biology; Internal medicine; Nuclear medicine; Cancer; Biochemistry","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0004801437,0.0004863648,0.0006209476,0.0003876348,0.0004924297,0.0003070795,0.0005083399,0.0004683341,0.001628315],"category_scores_gemma":[0.0003195601,0.0003023746,0.0004623199,0.0004369279,0.0002033729,0.0004396405,0.0002464698,0.0004787023,0.0007566517],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0004861789,"about_ca_system_score_gemma":0.0006456102,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.001577809,"about_ca_topic_score_gemma":0.001986893,"domain_scores_codex":[0.9997382,0.00006551117,0.00002879641,0.00005382761,0.00004820155,0.00006548531],"domain_scores_gemma":[0.9998509,0.0000269272,0.00003150493,0.00002225072,0.00003066198,0.00003778451],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0007225695,0.000119203,0.0001472801,0.0001587451,0.00003322857,0.0002401817,0.00007221954,0.001026828,0.9902716,0.0003478286,0.0002137918,0.006646584],"study_design_scores_gemma":[0.000134753,0.001328096,0.0005154635,0.000008048213,0.00007372293,0.0005401213,0.00002468391,0.0007881798,0.9859595,0.00006120109,0.01054537,0.00002100927],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.934122,0.01163611,0.04022975,0.0004247922,0.000230675,0.0008038841,0.00266923,0.0002802958,0.009603102],"genre_scores_gemma":[0.967693,0.004033546,0.02036926,0.00009892532,0.00004840547,0.0002046938,0.002300362,0.000129962,0.005121878],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.001628315,"threshold_uncertainty_score":0.005447209,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.08327797894450965,"score_gpt":0.387989811950493,"score_spread":0.3047118330059834,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}