{"id":"W2790192464","doi":"10.1002/pep2.24056","title":"New directions for urotensin II receptor ligands","year":2018,"lang":"en","type":"article","venue":"Peptide Science","topic":"Cardiovascular, Neuropeptides, and Oxidative Stress Research","field":"Medicine","cited_by":12,"is_retracted":false,"has_abstract":true,"ca_institutions":"Institut National de la Recherche Scientifique","funders":"Institute of Circulatory and Respiratory Health; Natural Sciences and Engineering Research Council of Canada","keywords":"Urotensin-II; Allosteric regulation; G protein-coupled receptor; Peptide; Receptor; Endogeny; Chemistry; Pharmacology; Biochemistry; Stereochemistry; Biology","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"codex-gemma-dda1882f352a","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0007066645,0.0001303447,0.0002351262,0.0002677928,0.0008710977,0.00008171823,0.0002594762,0.00003609034,0.0003108015],"category_scores_gemma":[0.001654633,0.0001075527,0.0002006083,0.001190263,0.001030331,0.0002325982,0.0001819281,0.000151067,0.0002270875],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0000919112,"about_ca_system_score_gemma":0.0006377795,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.000136664,"about_ca_topic_score_gemma":0.00003904056,"domain_scores_codex":[0.997999,0.00001783453,0.0001758734,0.0005590494,0.000722057,0.0005261686],"domain_scores_gemma":[0.9980793,0.000074651,0.00003778604,0.0005395973,0.000830336,0.0004383269],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"not_applicable","study_design_scores_codex":[0.0002185254,0.00007661538,0.001231785,0.00003029298,0.00005562356,0.000009031181,0.0007222343,0.00000205867,0.7763152,0.0005213763,0.09941595,0.1214013],"study_design_scores_gemma":[0.001021602,0.0009733476,0.02272039,0.00008812627,0.00004249037,0.00006893332,0.0001028442,0.00021576,0.4345238,0.0001227676,0.5399482,0.0001717464],"study_design_candidate":"bench_or_experimental","study_design_consensus":null,"genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.8687236,0.0007378554,0.01512132,0.005353265,0.002076421,0.001992902,0.00004355676,0.0003686152,0.1055824],"genre_scores_gemma":[0.9041877,0.0002321261,0.02114844,0.0006579196,0.002782947,0.00004894454,0.000009523777,0.00004142792,0.07089094],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.4405322,"threshold_uncertainty_score":0.6699867,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.03417980003985432,"score_gpt":0.3381726141962397,"score_spread":0.3039928141563854,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}