{"id":"W2790192464","doi":"10.1002/pep2.24056","title":"New directions for urotensin II receptor ligands","year":2018,"lang":"en","type":"article","venue":"Peptide Science","topic":"Cardiovascular, Neuropeptides, and Oxidative Stress Research","field":"Medicine","cited_by":12,"is_retracted":false,"has_abstract":true,"ca_institutions":"Institut National de la Recherche Scientifique","funders":"Institute of Circulatory and Respiratory Health; Natural Sciences and Engineering Research Council of Canada","keywords":"Urotensin-II; Allosteric regulation; G protein-coupled receptor; Peptide; Receptor; Endogeny; Chemistry; Pharmacology; Biochemistry; Stereochemistry; Biology","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0008649894,0.0004640836,0.0008058486,0.0006046027,0.0001578502,0.001027596,0.0006657426,0.0009464537,0.006032702],"category_scores_gemma":[0.0005242592,0.0001837646,0.0004412378,0.0004820734,0.0004137574,0.001468517,0.0006705796,0.002299373,0.002598052],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.00046555,"about_ca_system_score_gemma":0.0006798335,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0003223615,"about_ca_topic_score_gemma":0.0005582923,"domain_scores_codex":[0.9997891,0.0000600953,0.00002048828,0.00004354744,0.00004973919,0.00003713835],"domain_scores_gemma":[0.9997756,0.00008684202,0.00002662078,0.00001085891,0.00006710523,0.00003310173],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"design_other","study_design_gemma":"not_applicable","study_design_scores_codex":[0.0008140334,0.0002908266,0.0004713111,0.01235455,0.0001546902,0.0008477017,0.000218129,0.001409172,0.03883436,0.0435894,0.04219495,0.8588209],"study_design_scores_gemma":[0.0001113345,0.0006801681,0.0005027658,0.0012752,0.0001012931,0.0009458882,0.00009363033,0.0005007254,0.004828439,0.008118741,0.9828083,0.00003355233],"study_design_candidate":"not_applicable","study_design_consensus":null,"genre_codex":"review","genre_gemma":"empirical","genre_scores_codex":[0.002351407,0.9846827,0.00362353,0.002964788,0.001128197,0.00002908011,0.0001332407,0.00008071308,0.005006364],"genre_scores_gemma":[0.01893864,0.9679088,0.002853979,0.003098482,0.001146535,0.00008176463,0.0002859301,0.00002481065,0.005661014],"genre_candidate":"empirical","genre_consensus":null,"teacher_disagreement_score":0.006032702,"threshold_uncertainty_score":0.02018142,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.03417980003985432,"score_gpt":0.3381726141962397,"score_spread":0.3039928141563854,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}