{"id":"W3193528876","doi":"10.1002/ddr.21865","title":"Ketotifen is a Prodrug. Norketotifen is the active metabolite.","year":2021,"lang":"en","type":"article","venue":"Drug Development Research","topic":"Inflammatory mediators and NSAID effects","field":"Medicine","cited_by":4,"is_retracted":false,"has_abstract":true,"ca_institutions":"The Scarborough Hospital; Nucro Technics","funders":"","keywords":"Ketotifen; Metabolite; Pharmacology; Prodrug; Active metabolite; In vivo; Chemistry; Medicine; Internal medicine; Biology; Biochemistry","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0001190032,0.0004314024,0.0002432145,0.0004650989,0.0002001903,0.0002673997,0.0001616734,0.0003142584,0.003146848],"category_scores_gemma":[0.000151807,0.0001405604,0.0002386739,0.000252689,0.0002024517,0.000239632,0.0001890448,0.0003638193,0.001562837],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.000412693,"about_ca_system_score_gemma":0.0003152262,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0006935548,"about_ca_topic_score_gemma":0.001383776,"domain_scores_codex":[0.9998673,0.00001914549,0.00001449932,0.00002599164,0.00005313461,0.00001977308],"domain_scores_gemma":[0.9999089,0.00001082988,0.00003183198,0.000005518922,0.0000186549,0.00002417362],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0009793106,0.0001485631,0.001678874,0.0008922121,0.00003389329,0.0008108087,0.00003649852,0.0003439504,0.9219526,0.0008357596,0.001076803,0.07121085],"study_design_scores_gemma":[0.00006257476,0.002375,0.004720588,0.00004508187,0.0000393539,0.004325904,0.0000369444,0.0002394505,0.9217725,0.0001500253,0.06621561,0.00001706829],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.7808749,0.1219799,0.02863265,0.001200864,0.0009012932,0.0007172239,0.007950692,0.0006347995,0.05710768],"genre_scores_gemma":[0.9492191,0.02085067,0.009455133,0.0002265176,0.00007202542,0.0001315237,0.003219321,0.00002388056,0.01680183],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.003146848,"threshold_uncertainty_score":0.01052731,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.05725537217089694,"score_gpt":0.3666357999871766,"score_spread":0.3093804278162797,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}