{"id":"W3193528876","doi":"10.1002/ddr.21865","title":"Ketotifen is a Prodrug. Norketotifen is the active metabolite.","year":2021,"lang":"en","type":"article","venue":"Drug Development Research","topic":"Inflammatory mediators and NSAID effects","field":"Medicine","cited_by":4,"is_retracted":false,"has_abstract":true,"ca_institutions":"The Scarborough Hospital; Nucro Technics","funders":"","keywords":"Ketotifen; Metabolite; Pharmacology; Prodrug; Active metabolite; In vivo; Chemistry; Medicine; Internal medicine; Biology; Biochemistry","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"codex-gemma-dda1882f352a","candidate_categories":["insufficient_payload"],"consensus_categories":["insufficient_payload"],"category_scores_codex":[0.003168681,0.0002551515,0.0004157121,0.0002499015,0.0006104161,0.0001062106,0.0003220138,0.0001185828,0.001618447],"category_scores_gemma":[0.0006991535,0.0001655302,0.0001377614,0.001215229,0.0002130298,0.0001184534,0.0004118886,0.001015071,0.001594336],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0002893237,"about_ca_system_score_gemma":0.002876169,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.00003129125,"about_ca_topic_score_gemma":0.00002463698,"domain_scores_codex":[0.9955373,0.0005387792,0.0003920177,0.0006450716,0.001927436,0.0009594177],"domain_scores_gemma":[0.9971257,0.0005247008,0.0000613979,0.0007835981,0.001139636,0.0003649589],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"not_applicable","study_design_gemma":"not_applicable","study_design_scores_codex":[0.001311101,0.001169897,0.05861242,0.001560481,0.001958463,0.002330303,0.1822007,0.000001225222,0.01854714,0.001054831,0.4013252,0.3299282],"study_design_scores_gemma":[0.0007225875,0.0000204321,0.05904947,0.0001226103,0.00002792957,0.00004290307,0.001964781,0.00003300382,0.4059448,0.00007159779,0.531832,0.0001678293],"study_design_candidate":"not_applicable","study_design_consensus":"not_applicable","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9592373,0.001347019,0.000008221566,0.01975505,0.0003334109,0.00127771,0.00001225746,0.00006846968,0.01796059],"genre_scores_gemma":[0.8579143,0.0004851097,0.001627108,0.004266753,0.0008838808,0.0006727013,0.0001104557,0.00009789957,0.1339418],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.3873977,"threshold_uncertainty_score":0.9992942,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.05725537217089694,"score_gpt":0.3666357999871766,"score_spread":0.3093804278162797,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}