{"id":"W4400201615","doi":"10.3390/molecules29133102","title":"Synthesis and Evaluation of the First 68Ga-Labeled C-Terminal Hydroxamate-Derived Gastrin-Releasing Peptide Receptor-Targeted Tracers for Cancer Imaging with Positron Emission Tomography","year":2024,"lang":"en","type":"article","venue":"Molecules","topic":"Neuropeptides and Animal Physiology","field":"Neuroscience","cited_by":2,"is_retracted":false,"has_abstract":true,"ca_institutions":"University of British Columbia; Terry Fox Research Institute","funders":"Canadian Institutes of Health Research; University of British Columbia; China Scholarship Council","keywords":"Biodistribution; Chemistry; Gastrin; Positron emission tomography; Peptide; In vivo; Antagonist; Pancreas; Nuclear medicine; Receptor; Molecular biology; Medicine; Biochemistry; In vitro; Biology","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.000387066,0.0005075001,0.0003920218,0.0002554929,0.0001764929,0.0002887881,0.0004626358,0.0005640496,0.000653133],"category_scores_gemma":[0.0003028114,0.0002476736,0.0003077211,0.0002441406,0.0002262628,0.0002608494,0.0002169905,0.0004097621,0.0004521589],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0005501917,"about_ca_system_score_gemma":0.0004195527,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.001444721,"about_ca_topic_score_gemma":0.001999358,"domain_scores_codex":[0.9998606,0.00003687996,0.00001079989,0.00002338613,0.00003834895,0.00002984848],"domain_scores_gemma":[0.9998771,0.00001622879,0.00002231648,0.00001039842,0.00003268691,0.00004129704],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0001476492,0.00004395592,0.00006438645,0.00009831514,0.000008097049,0.00006409489,0.00003035084,0.0003779752,0.9959928,0.0001934476,0.00007562976,0.00290322],"study_design_scores_gemma":[0.0000889006,0.001785861,0.0007777028,0.00001204103,0.00003578793,0.0002794986,0.00002356287,0.002014907,0.98844,0.00004764769,0.006474596,0.00001950073],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9679605,0.007710948,0.01997559,0.0001698303,0.00006369347,0.00082148,0.0005656264,0.0001608766,0.00257146],"genre_scores_gemma":[0.9406543,0.005679022,0.04724677,0.0002346609,0.00003450323,0.0006191965,0.001425026,0.00007873232,0.004027857],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.001444721,"threshold_uncertainty_score":0.003991961,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.01876457480755407,"score_gpt":0.2652596203392088,"score_spread":0.2464950455316547,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}