{"id":"W4401658384","doi":"10.1021/acs.molpharmaceut.4c00549","title":"First-Generation Radiolabeled Cyclic Peptides for Molecular Imaging of Platelet-Derived Growth Factor Receptor α","year":2024,"lang":"en","type":"article","venue":"Molecular Pharmaceutics","topic":"Radiopharmaceutical Chemistry and Applications","field":"Medicine","cited_by":1,"is_retracted":false,"has_abstract":true,"ca_institutions":"University of Alberta","funders":"","keywords":"Chemistry; Cyclic peptide; Receptor; Biophysics; Pharmacology; Cancer research; Biochemistry; Medicine; Peptide; Biology","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"codex-gemma-dda1882f352a","candidate_categories":["metaepi_narrow"],"consensus_categories":[],"category_scores_codex":[0.0001491222,0.0002808053,0.0003423154,0.0001060464,0.0001005035,0.00005536106,0.0001567051,0.0001123996,0.0001266893],"category_scores_gemma":[0.000129918,0.0002789279,0.000282255,0.0003515284,0.0001202455,0.00008968044,0.00003660521,0.0003090412,0.00002312014],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.000113983,"about_ca_system_score_gemma":0.0001069628,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.000002919661,"about_ca_topic_score_gemma":1.527391e-7,"domain_scores_codex":[0.9983919,0.00003526001,0.0004502164,0.0004645031,0.0002893304,0.0003687702],"domain_scores_gemma":[0.9990574,0.0001115667,0.00007759759,0.0002902233,0.0001944535,0.0002687948],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.00007608713,0.000119024,0.0001121739,0.0009893191,0.0002624767,0.00007098845,0.0001163452,0.000136205,0.9928831,0.001136195,0.0009716699,0.003126422],"study_design_scores_gemma":[0.001262908,0.000044234,0.00001676575,0.0001107748,0.0003250514,0.00006442214,0.00001668006,0.070248,0.8972587,0.000168317,0.0302472,0.0002369221],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9201109,0.006185033,0.06684302,0.004686701,0.0002457404,0.001169549,0.0001662445,0.0002237039,0.0003691324],"genre_scores_gemma":[0.9907389,0.0004180436,0.007017721,0.0009494752,0.0002513434,0.0001890569,0.0002508427,0.00008409264,0.0001005118],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.09562437,"threshold_uncertainty_score":0.9999663,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.03980676152551487,"score_gpt":0.3446536814110301,"score_spread":0.3048469198855152,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}