{"id":"W4403869318","doi":"10.2139/ssrn.4987379","title":"Diamino Variants of Piperazine-Based Tissue Transglutaminase Inhibitors","year":2024,"lang":"en","type":"preprint","venue":"SSRN Electronic Journal","topic":"Blood properties and coagulation","field":"Medicine","cited_by":0,"is_retracted":false,"has_abstract":false,"ca_institutions":"University of Ottawa","funders":"","keywords":"Tissue transglutaminase; Piperazine; Chemistry; Pharmacology; Biochemistry; Enzyme; Medicine; Organic chemistry","routes":{"ca_aff":true,"ca_fund":false,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0001598305,0.0003023942,0.0002248979,0.00009627963,0.00008086617,0.0002067457,0.0003534925,0.000229281,0.002609057],"category_scores_gemma":[0.0001856138,0.00009272772,0.0001381769,0.0001222045,0.0001549466,0.0002675244,0.0001978562,0.0006543891,0.0006761157],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.000201165,"about_ca_system_score_gemma":0.00008406511,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0002170935,"about_ca_topic_score_gemma":0.0003043169,"domain_scores_codex":[0.9999065,0.00002536249,0.000007233474,0.00002021006,0.00002274138,0.00001778222],"domain_scores_gemma":[0.9999278,0.00001101984,0.00002704001,0.000009841374,0.000009248183,0.00001507201],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0009556346,0.00007483038,0.0001832091,0.000193969,0.00003953179,0.0002658291,0.00004418215,0.001040963,0.9777853,0.002818863,0.0007662193,0.01583142],"study_design_scores_gemma":[0.0001717694,0.003050773,0.001052181,0.0000219553,0.00006884789,0.001632136,0.00003477342,0.004090053,0.9565917,0.0007228762,0.03253832,0.00002467492],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.946305,0.01289961,0.01981721,0.0007730733,0.0003646158,0.0001104706,0.000480802,0.0003486042,0.0189006],"genre_scores_gemma":[0.9821367,0.002871116,0.006255215,0.0001872169,0.00004868799,0.00003302967,0.0003492818,0.0000319139,0.008086894],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.002609057,"threshold_uncertainty_score":0.008728147,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.01131050554836648,"score_gpt":0.2584139302181401,"score_spread":0.2471034246697736,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}