{"id":"W4408790789","doi":"10.3390/ph18040449","title":"Novel 177Lu-Labeled [Thz14]Bombesin(6–14) Derivatives with Low Pancreas Accumulation for Targeting Gastrin-Releasing Peptide Receptor-Expressing Cancer","year":2025,"lang":"en","type":"article","venue":"Pharmaceuticals","topic":"Neuropeptides and Animal Physiology","field":"Neuroscience","cited_by":2,"is_retracted":false,"has_abstract":true,"ca_institutions":"University of British Columbia; Terry Fox Research Institute","funders":"Canadian Institutes of Health Research; University of British Columbia; China Scholarship Council","keywords":"Bombesin; Biodistribution; DOTA; Chemistry; Radionuclide therapy; Gastrin; Pancreas; In vivo; Cancer research; Nuclear medicine; Medicine; Receptor; In vitro; Biochemistry; Biology","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"codex-gemma-dda1882f352a","candidate_categories":["metaepi_narrow"],"consensus_categories":[],"category_scores_codex":[0.0001672343,0.0003369664,0.0004089964,0.0001143135,0.0005086335,0.000157065,0.0003009691,0.0000729275,0.0001144986],"category_scores_gemma":[0.000970957,0.0002858625,0.0001022039,0.0004971752,0.0002451135,0.0004216119,0.0001477813,0.0003287961,0.00001750504],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.00008578062,"about_ca_system_score_gemma":0.0001344579,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.00002403796,"about_ca_topic_score_gemma":0.000002348808,"domain_scores_codex":[0.9975848,0.0001772058,0.0004431565,0.0008175274,0.0002391162,0.0007382474],"domain_scores_gemma":[0.9981067,0.001152141,0.0002188453,0.0002040774,0.0001603284,0.0001579559],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0009178976,0.0001648262,0.0007944771,0.0001530585,0.00002530443,0.000002964364,0.00007771009,0.001065677,0.988319,0.001323476,0.0006536281,0.006501951],"study_design_scores_gemma":[0.002035736,0.0001180723,0.001723294,0.0004101317,0.00006519404,0.000004076552,0.00004985568,0.008744899,0.9664684,0.0002334404,0.01980748,0.0003394484],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9877341,0.0002016268,0.008928025,0.0007309103,0.0003403169,0.0008631806,0.00006292974,0.0002028429,0.0009360674],"genre_scores_gemma":[0.9904738,0.0001813555,0.005267008,0.003142657,0.0002754225,0.0001387425,0.0000093918,0.00005843334,0.0004531545],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.02185066,"threshold_uncertainty_score":0.9999593,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.1029642103078166,"score_gpt":0.4008433594543915,"score_spread":0.2978791491465749,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}