{"id":"W4415827410","doi":"10.1016/j.bmc.2025.118476","title":"Tissue transglutaminase inhibitors over the past decade","year":2025,"lang":"en","type":"article","venue":"Bioorganic & Medicinal Chemistry","topic":"Blood properties and coagulation","field":"Medicine","cited_by":1,"is_retracted":false,"has_abstract":true,"ca_institutions":"University of Ottawa","funders":"Natural Sciences and Engineering Research Council of Canada","keywords":"Tissue transglutaminase; Enzyme; Intracellular; Enzyme inhibitor; Fibrosis; In vitro","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"codex-gemma-dda1882f352a","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0001713657,0.0001807389,0.000236507,0.00002716121,0.0001285434,0.00001629628,0.0001535028,0.0001766771,0.0008296563],"category_scores_gemma":[0.00008044521,0.0001129357,0.00007198367,0.0003441492,0.0001658645,0.00003194297,0.0000408028,0.0003386723,0.00002413418],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.00008022431,"about_ca_system_score_gemma":0.000184837,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.00005015787,"about_ca_topic_score_gemma":0.000002895905,"domain_scores_codex":[0.9988629,0.00001695573,0.0002876061,0.0002670617,0.0003190272,0.0002464782],"domain_scores_gemma":[0.9993378,0.00004281509,0.00005546813,0.000378621,0.00006539142,0.000119929],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"bench_or_experimental","study_design_gemma":"bench_or_experimental","study_design_scores_codex":[0.0001678454,0.0001250535,0.006609383,0.0004769746,0.0001057381,0.00004366705,0.0002939168,2.924669e-7,0.935836,0.00003749963,0.02128274,0.0350209],"study_design_scores_gemma":[0.001567834,0.00008563086,0.03931965,0.0004036756,0.0004368308,0.0001171863,0.000691269,0.00003376229,0.8505359,0.00004993391,0.1066089,0.0001495158],"study_design_candidate":"bench_or_experimental","study_design_consensus":"bench_or_experimental","genre_codex":"empirical","genre_gemma":"empirical","genre_scores_codex":[0.9725961,0.004533722,0.0001719021,0.01427172,0.0002579527,0.0002577691,0.000003892623,0.00008731819,0.007819589],"genre_scores_gemma":[0.9903505,0.00008000463,0.00003166587,0.001787585,0.0009042367,0.00001535056,0.00002261629,0.00001901484,0.006789037],"genre_candidate":"empirical","genre_consensus":"empirical","teacher_disagreement_score":0.08532611,"threshold_uncertainty_score":0.9084155,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.008772836132755703,"score_gpt":0.2537163432516543,"score_spread":0.2449435071188986,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}