{"id":"W4415827410","doi":"10.1016/j.bmc.2025.118476","title":"Tissue transglutaminase inhibitors over the past decade","year":2025,"lang":"en","type":"article","venue":"Bioorganic & Medicinal Chemistry","topic":"Blood properties and coagulation","field":"Medicine","cited_by":1,"is_retracted":false,"has_abstract":true,"ca_institutions":"University of Ottawa","funders":"Natural Sciences and Engineering Research Council of Canada","keywords":"Tissue transglutaminase; Enzyme; Intracellular; Enzyme inhibitor; Fibrosis; In vitro","routes":{"ca_aff":true,"ca_fund":true,"ca_venue":false,"about_ca":false,"invisible_to_affiliation_only":false},"retraction":null,"screen":null,"direct_labels":[],"prediction":{"model_version":"metacan-v3-hybrid-931329e0061c","candidate_categories":[],"consensus_categories":[],"category_scores_codex":[0.0006468753,0.0007163453,0.0006021744,0.0006884637,0.0001718809,0.0006191154,0.0003661626,0.0005937916,0.003453277],"category_scores_gemma":[0.0007772637,0.0002036839,0.0003238941,0.0007882719,0.0002045949,0.0007415917,0.0004333749,0.001724618,0.001597588],"about_ca_system_candidate":false,"about_ca_system_consensus":false,"about_ca_system_score_codex":0.0004758956,"about_ca_system_score_gemma":0.0004679907,"about_ca_topic_candidate":false,"about_ca_topic_consensus":false,"about_ca_topic_score_codex":0.0004913121,"about_ca_topic_score_gemma":0.001055013,"domain_scores_codex":[0.9997877,0.00003550162,0.00002537544,0.00005023011,0.00007190823,0.00002925111],"domain_scores_gemma":[0.9997391,0.00006903954,0.00004750791,0.000008835239,0.00009230022,0.0000432385],"domain_codex":null,"domain_gemma":null,"domain_candidate":null,"domain_consensus":null,"study_design_codex":"design_other","study_design_gemma":"not_applicable","study_design_scores_codex":[0.0005383295,0.0002851936,0.0004507554,0.008727329,0.0002765349,0.000473217,0.0001381372,0.001304387,0.03518626,0.006634932,0.05797347,0.8880115],"study_design_scores_gemma":[0.00006482799,0.0006756401,0.0005621854,0.0005653548,0.0001502176,0.001188673,0.00002765693,0.0003050631,0.0136344,0.0008313297,0.9819703,0.0000242993],"study_design_candidate":"not_applicable","study_design_consensus":null,"genre_codex":"review","genre_gemma":"review","genre_scores_codex":[0.003362934,0.9867742,0.002174759,0.001231461,0.001180138,0.00002525588,0.0001315655,0.00006937501,0.005050317],"genre_scores_gemma":[0.01915351,0.9671856,0.001793009,0.002194465,0.0009731614,0.00005103504,0.0004404983,0.00001913334,0.008189456],"genre_candidate":"review","genre_consensus":"review","teacher_disagreement_score":0.003453277,"threshold_uncertainty_score":0.01155239,"prediction_status":"machine_predicted_unvalidated"},"machine_scores":{"provisional":true,"baseline":true,"maturity_gate_passed":false,"score_opus":0.008772836132755703,"score_gpt":0.2537163432516543,"score_spread":0.2449435071188986,"validation_status":"score_only:v0-immature-baseline","note":"Baseline scores from an immature model (maturity gate not passed). Scores rank; they never assert a category."}}