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Record W7005790532

Single-nucleus profiling of the human brain to identify therapeutic targets

2023· other· en· W7005790532 on OpenAlex

Why this work is in the frame

A frame that forgets how it found something cannot be audited. These are the routes that admitted this work.

fundA Canadian funder is recorded on the work.
no affNo Canadian affiliation: this work is invisible to an affiliation-only frame.
No Canadian affiliation. An affiliation-only frame, the usual design, would never have seen this work. It is one of the works that make the case for inverting the frame.

Bibliographic record

VenueeScholarship (California Digital Library) · 2023
Typeother
Languageen
FieldMedicine
TopicMedicinal Plant Extracts Effects
Canadian institutionsnot available
FundersNational Institute of General Medical SciencesNational Institutes of HealthUniversity of California, San DiegoDalhousie UniversityShaffer Family FoundationGoizueta Business School, Emory UniversityUniversity of WashingtonEmory UniversityUniversity of MiamiU.S. Department of Defense
KeywordsProfiling (computer programming)Human brainHuman studiesDrug developmentHuman useDrug discovery
DOInot available

Abstract

fetched live from OpenAlex

The human brain is underpinned by a massive cellular complexity. A diverse conglomerate of cells, over 100 billion of them, functionally interact to power the most uniquely human organ. Unfortunately, the brain often encounters difficulties, and these neurological disorders drive significant clinical challenges. Most neurological disorders have no consistently effective therapeutic treatments. The work of this dissertation has been conducted with a single goal in mind: to improve the understanding of the human brain, in turn enabling the development of effective therapeutics to treat neurological disorders. To accomplish this, we conducted method development to enable effective single-nucleus profiling of the human brain, outlined tools for analyzing this data, carefully selected targets that may drive functional improvements, and developed and tested therapeutics capable of changing the brain. Here, we have profiled human brains with Down syndrome and matched controls to identify microglial overactivation, and a unique transcription factor, RUNX1, that appear to drive memory deficits. Additionally, we show that a potential therapeutic, targeting RUNX1, can reverse certain aspects of this biology. This work establishes a foundation for drug discovery, utilizing single-nucleus RNA-sequencing data to guide target selection and providing conceptual proof that these efforts can yield efficacious therapeutics.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.001
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesMeta-epidemiology (narrow), Insufficient payload (model declined to judge)
Consensus categoriesInsufficient payload (model declined to judge)
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Not applicable · Consensus signal: Not applicable
GenreCandidate signal: Other · Consensus signal: Other
Teacher disagreement score0.309
Threshold uncertainty score1.000

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0000.001
Meta-epidemiology (narrow)0.0010.000
Meta-epidemiology (broad)0.0010.000
Bibliometrics0.0010.001
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0010.000
Research integrity0.0010.001
Insufficient payload (model declined to judge)0.0010.003

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.028
GPT teacher head0.282
Teacher spread0.253 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it