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Record W1991205167 · doi:10.1055/s-2009-1216535

Antitumor Activity of Aralia racemosa

2009· article· en· W1991205167 on OpenAlexfundno aff
JA Clement, TJ Willis, RM Kelly, JA McCoy, JD Schmitt

Bibliographic record

VenuePlanta Medica · 2009
Typearticle
Languageen
FieldAgricultural and Biological Sciences
TopicPlant Pathogens and Resistance
Canadian institutionsnot available
FundersNational Institute on Drug AbuseAgricultural Research ServiceUniversity of British ColumbiaUniversity of Illinois at Urbana-ChampaignChinese Academy of SciencesKurukshetra UniversityUniversity of Illinois at ChicagoNational Oceanic and Atmospheric AdministrationU.S. Food and Drug AdministrationNational Science Foundation of Sri LankaUniversity of ColomboU.S. Department of AgricultureWestern Carolina UniversityInternational Science CouncilNational Center for Complementary and Alternative MedicineChina Academy of Traditional Chinese MedicineNational Institutes of HealthNational Center for Research ResourcesNational Institute of Allergy and Infectious DiseasesTürkiye Bilimsel ve Teknolojik Araştırma KurumuHong Kong Polytechnic UniversityNational Science FoundationDeutsche KrebshilfeNational Natural Science Foundation of ChinaTata TrustsUniversity Grants CommissionWake Forest University
KeywordsBioassayCytotoxic T cellTerpenoidFractionationHigh-performance liquid chromatographyTraditional medicineCytotoxicityBiologyChemistryBotanyIn vitroChromatographyBiochemistryMedicineEcology

Abstract

fetched live from OpenAlex

The southern Appalachians are home to an extraordinary variety of plant species, many of which have been used medicinally by local populations. The vast majority of these species have not been studied for their antitumor activity, constituting a significant bioexploration opportunity. We have recently begun a targeted screening program for identifying plants indigenous to Western North Carolina with potential antitumor activity. Initial screening against the MCF-7 breast tumor cell line identified an extract of Aralia racemosa (aerial parts) as having cytotoxic activity. Combined CH 2 Cl 2 extractions of the acidified crude organic extract showed dose-dependent toxicity towards MCF-7 cells, with IC 50 around 100 µg/mL. Bioassay-guided fractionation by reverse phase C 18 open column chromatography, followed by reverse phase C 18 HPLC, afforded the major cytotoxic component, a twenty-carbon terpenoid, along with an inactive twenty-carbon compound. The major cytotoxic compound gives 73% inhibition growth of MCF-7 cells at 100 µg/mL. The structure has been characterized by NMR spectroscopy and ESI-MS, and these results will be presented. Acknowledgements: We thank the Western Carolina University SURF Program for summer support for T.J.W. We thank Wake Forest University Health Sciences Virus and Vector Core Laboratory for assay work.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame machine prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. The Gemma side is a direct model label for every work in the frame, read from the title-only record. The Codex side is a classifier learned from the 10,348 direct Codex labels and calibrated to design-weighted sample rates; fields without enough sample support carry no Codex call. Candidate is the union of the two sides; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.000
Version: metacan-v3-hybrid-931329e0061cValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.002
Threshold uncertainty score0.008

Distilled classifier scores by category (both heads)

CategoryCodexGemma
Metaresearch0.0000.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0020.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.016
GPT teacher head0.218
Teacher spread0.202 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one source (direct Gemma or distilled Codex), not a consensus.

The models applied no category: nothing in the taxonomy fit this work.
Study designBench or experimental
Domainnot available
GenreEmpirical

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations4
Published2009
Admission routes1
Has abstractyes

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