MétaCan
Menu
Back to cohort
Record W2049896452 · doi:10.1021/jp993406a

A Volumetric Study of Cyclodextrin-α,ω-Alkyl Dicarboxylate Anion Complexes in Aqueous Solutions

2000· article· en· W2049896452 on OpenAlexafffund
Lee D. Wilson, Ronald E. Verrall

Bibliographic record

VenueThe Journal of Physical Chemistry B · 2000
Typearticle
Languageen
FieldPharmacology, Toxicology and Pharmaceutics
TopicDrug Solubulity and Delivery Systems
Canadian institutionsSteacie Institute for Molecular SciencesUniversity of Saskatchewan
FundersNatural Sciences and Engineering Research Council of Canada
KeywordsAqueous solutionChemistryTernary operationAlkylMethyleneCyclodextrinHomologous seriesMoleculeCrystallographyCarboxylateDilutionMolar volumeMedicinal chemistryInorganic chemistryStereochemistryOrganic chemistryThermodynamics

Abstract

fetched live from OpenAlex

The apparent molar volumes ( V φ,S ) of a homologous series of sodium α,ω-alkyl dicarboxylate [(CH 2 ) x (CO 2 Na) 2, x = 4, 6, 8, 10, 12] salts (S) have been determined in water (w) and in aqueous cyclodextrin (CD) solutions at 25 °C. The magnitude of V φ,S in ternary (w+S+CD) solutions containing β-CD and DM-β-CD (2,6-di-O-methyl β-cyclodextrin) are greater than in the binary (w+S) aqueous systems. However, in ternary solutions containing α-CD, the magnitude of V φ,S is lower than in the binary systems. The apparent molar volume (AMV) of the α,ω-alkyl dicarboxylate salts in ternary aqueous solutions can be related to the formation of inclusion complexes between the CD and the anions (C x 2- where x = 6, 8, 10, 12). The transfer volume of the C x 2- guests at infinite dilution from water to aqueous CD solutions are well described by a simple molecular additivity scheme which accounts for the number of methylene groups of the guest that are included and the number of water molecules displaced from the CD interior. The volumetric properties of the ternary systems have been quantitatively described in terms of a two- or three-site model that accounts for the AMV of bound and unbound species. In cases where CD-S inclusion complexes are formed, β-CD and DM-β-CD form 1:1, α-CD forms 1:1 ( x ≤ 8) and 2:1 complexes ( x ≥ 10). The binding mode involves threading of the methylene chain of the guest through the CD interior while the carboxylate groups remain hydrated in the bulk solvent or adjacent to the CD annuli. The calculated 1:1 binding constants ( K 1:1 ) vary between 10 1 −10 3 kg mol -1 and the 2:1 binding constants ( K 2:1 ) are ca. 10 2 kg 2 mol -2 . The relative binding affinity of the host systems with a common C x 2- guest are as follows: α-CD > β-CD > DM-β-CD, and these differences are mainly related to the diameter of the host cavity.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.001
metaresearch head score (Gemma)0.000
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: none
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.397
Threshold uncertainty score0.475

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0010.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.001
Insufficient payload (model declined to judge)0.0000.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.081
GPT teacher head0.387
Teacher spread0.306 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one teacher head, not a consensus.

The models applied no category: nothing in the taxonomy fit this work.
Study designBench or experimental
Domainnot available
GenreEmpirical

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations32
Published2000
Admission routes2
Has abstractyes

Explore more

Same venueThe Journal of Physical Chemistry BSame topicDrug Solubulity and Delivery SystemsFrench-language works237,207