MétaCan
Menu
Back to cohort
Record W2163300687 · doi:10.1002/ddr.10016

Gabapentin: A novel analgesic targeting voltage‐gated calcium channels

2001· article· en· W2163300687 on OpenAlex

Why this work is in the frame

A frame that forgets how it found something cannot be audited. These are the routes that admitted this work.

affAt least one author lists a Canadian institution in the pinned OpenAlex snapshot.
fundA Canadian funder is recorded on the work.

Bibliographic record

VenueDrug Development Research · 2001
Typearticle
Languageen
FieldMedicine
TopicPain Mechanisms and Treatments
Canadian institutionsUniversity of British Columbia
FundersCanadian Institutes of Health Research
KeywordsGabapentinAnticonvulsantPharmacologyCalcium channelChemistryVoltage-dependent calcium channelNeuroscienceNeurotransmitterNeuropathic painAnalgesicCalciumMechanism of actionReceptorEpilepsyMedicinePsychologyBiochemistry

Abstract

fetched live from OpenAlex

Abstract Given their vital roles in mediating neuronal excitability, it is not surprising that voltage‐gated calcium channels have been implicated in contributing to the development and maintenance of pain processes. Gabapentin, a synthetic analog of the neurotransmitter γ‐aminobutyric acid (GABA), is a clinically effective anticonvulsant recently shown to be efficacious also for a variety of neuropathic pain conditions. While its mechanism of action is incompletely understood, current evidence suggests that gabapentin does not directly interact with GABA receptors but rather modulates the activity of high threshold calcium channels. Although gabapentin binds to the calcium channel α2δ ancillary subunit, it remains to be determined whether this interaction solely accounts for its therapeutic effects. Drug Dev. Res. 54:167–172, 2002. © 2002 Wiley‐Liss, Inc.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.003
metaresearch head score (Gemma)0.000
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesInsufficient payload (model declined to judge)
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: none
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.514
Threshold uncertainty score1.000

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0030.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0010.001
Science and technology studies0.0010.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.001
Insufficient payload (model declined to judge)0.0010.001

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.115
GPT teacher head0.383
Teacher spread0.269 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it