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Record W2164260704 · doi:10.1109/bibm.2009.60

Neural Grammar Networks in QSAR Chemistry

2009· article· en· W2164260704 on OpenAlexafffund
Y. T. Eddie, Stefan C. Kremer

Bibliographic record

Venuenot available
Typearticle
Languageen
FieldComputer Science
TopicComputational Drug Discovery Methods
Canadian institutionsUniversity of Guelph
FundersNatural Sciences and Engineering Research Council of Canada
KeywordsQuantitative structure–activity relationshipParsingComputer scienceArtificial neural networkArtificial intelligenceGrammarString (physics)Machine learningRepresentation (politics)CheminformaticsNatural language processingTheoretical computer scienceMathematicsChemistry

Abstract

fetched live from OpenAlex

In this paper, we describe the neural grammar network (NGN) and its application to quantitative structure-activity relationship (QSAR) in computational chemistry. The NGN is a novel machine learning device that applies the generic function approximation capability of a dynamic recursive neural network to the syntactic structure of a parsed string. In our QSAR task, we represent each molecule by a formal string representation (SMILES and InChI), and utilize an NGN instance to associate each with a real-value that describes the degree of binding, inhibition or affinity a given molecule has with a target protein. We find that the NGN can on average outperform previous work in regression tasks, yielding performances of up to 0.79 (sd = 0.23) in predictive r-squared scores and up to 74.8 (sd = 1.63) percent concordance in classification tasks.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.000
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Simulation or modeling · Consensus signal: Simulation or modeling
GenreCandidate signal: Empirical · Consensus signal: none
Teacher disagreement score0.855
Threshold uncertainty score0.326

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0000.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0010.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0000.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.011
GPT teacher head0.271
Teacher spread0.260 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one teacher head, not a consensus.

The models applied no category: nothing in the taxonomy fit this work.
Study designSimulation or modeling
Domainnot available
GenreEmpirical

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations3
Published2009
Admission routes2
Has abstractyes

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