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Record W2166170098 · doi:10.1002/chem.201302959

Synthesis and Theoretical Investigation of a 1,8‐Bis(bis(diisopropylamino)cyclopropeniminyl)naphthalene Proton Sponge Derivative

2013· article· en· W2166170098 on OpenAlex

Why this work is in the frame

A frame that forgets how it found something cannot be audited. These are the routes that admitted this work.

affAt least one author lists a Canadian institution in the pinned OpenAlex snapshot.
fundA Canadian funder is recorded on the work.

Bibliographic record

VenueChemistry - A European Journal · 2013
Typearticle
Languageen
FieldChemistry
TopicSynthesis and Properties of Aromatic Compounds
Canadian institutionsBrock University
FundersBrock UniversityMcMaster UniversityRyerson University
KeywordsProtonationNaphthaleneChemistryProtonDerivative (finance)AromaticitySpongeCrystal structureProton affinityComputational chemistryProton NMRCrystallographyStereochemistryMedicinal chemistryMoleculeOrganic chemistryIon

Abstract

fetched live from OpenAlex

We report herein the synthesis and characterization of a new proton sponge derivative, 1,8-bis(bis(diisopropylamino)cyclopropeniminyl)naphthalene 4 (DACN), as well as its bis-protonated counterpart 6. A crystal structure of 6 is presented, along with variable temperature (1)H NMR data on the BF4(-) salt (6⋅BF4). DFT calculations were performed to investigate the structure of the monoprotonated species 7 and to gain insight into the structural and electronic nature of all three species. The proton affinity (PA) of 4, calculated at the B3LYP/6-311G++(d,p)//B3LYP/6-31G(d,p) level, taking into account thermal corrections from the B3LYP/6-31G(d,p) method, was 282.3 kcal mol(-1), while its pKa was estimated at 27.0. NICS calculations were performed to examine the changes in aromaticity within these systems upon each successive protonation. Lastly, homodesmotic reaction schemes were used in order to estimate the factors contributing to the strong PA predicted for 4.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.001
metaresearch head score (Gemma)0.001
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesMeta-epidemiology (narrow), Insufficient payload (model declined to judge)
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.053
Threshold uncertainty score1.000

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0010.001
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.000
Science and technology studies0.0000.001
Scholarly communication0.0000.000
Open science0.0010.000
Research integrity0.0000.001
Insufficient payload (model declined to judge)0.0080.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.014
GPT teacher head0.194
Teacher spread0.180 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it