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Record W2230099494 · doi:10.1007/978-1-61779-213-7_6

Drug-Cytokine Interactions

2011· book-chapter· en· W2230099494 on OpenAlexaff
Jenna O. McNeil, Kerry B. Goralski

Bibliographic record

VenueHumana Press eBooks · 2011
Typebook-chapter
Languageen
FieldMedicine
TopicDrug Transport and Resistance Mechanisms
Canadian institutionsDalhousie University
Fundersnot available
KeywordsCytokineDrugPharmacologyImmune systemTumor necrosis factor alphaImmunologyDrug metabolismBiologyMedicineInflammation

Abstract

fetched live from OpenAlex

There are many documented examples of altered drug disposition in human conditions that stimulate host cytokine responses. These include viral, ­bacterial or parasitic infections, tissue injury, surgery, cancer and autoimmune ­conditions. Interferons, interleukins-1 and-6 and tumour necrosis factor are the central mediators. These cytokines have been traditionally viewed with respect to their ability to suppress hepatic cytochrome P450 (CYP)-mediated drug ­detoxification. Such aberrant drug handling has placed patients at risk for adverse drug responses to low therapeutic index, CYP-metabolized drugs like theophylline. It is now evident that drug-cytokine interactions are broader than once appreciated. They involve CYPs and drug transporter proteins like ABCB1 (P-glycoprotein) in the liver, intestine, kidney, blood-brain barrier, placenta and even immune cells. The consequences of drug-cytokine interactions are altered absorption, elimination and/or cellular and tissue distribution of drugs. The outcomes can be negative or positive depending on the drug, the anatomical site of the interaction and the therapeutic objectives. This chapter provides a historical overview of drug-cytokine ­interactions, discuss recent advances and examines the clinical scenarios in which infections or inflammation might lead to abnormal drug handling and drug responses.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.000
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesMeta-epidemiology (narrow), Insufficient payload (model declined to judge)
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Not applicable · Consensus signal: none
GenreCandidate signal: Other · Consensus signal: Other
Teacher disagreement score0.964
Threshold uncertainty score1.000

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0000.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0010.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.001
Insufficient payload (model declined to judge)0.0020.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.074
GPT teacher head0.271
Teacher spread0.196 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one teacher head, not a consensus.

Study designNot applicable
Domainnot available
GenreOther

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations6
Published2011
Admission routes1
Has abstractyes

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